SOLID-PHASE PHOSPHORYLATION OF A PEPTIDE BY THE H-PHOSPHONATE METHOD

被引：22

作者：

LARSSON, E ^{[1
]}

LUNING, B ^{[1
]}

机构：

[1] UNIV STOCKHOLM,DEPT ORGAN CHEM,S-10691 STOCKHOLM,SWEDEN

来源：

TETRAHEDRON LETTERS | 1994年 / 35卷 / 17期

关键词：

D O I：

10.1016/S0040-4039(00)77019-5

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The partially protected peptide SerValSerGluAla was selectively phosphorylated at Ser3 by benzyl H-phosphonate activated by pivaloyl chloride in pyridine, followed by in situ oxidation with iodine.

引用

页码：2737 / 2738

页数：2

共 6 条

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[2]

GAREGG PJ, 1985, CHEM SCRIPTA, V25, P280

[3]

GAREGG PJ, 1986, CHEM SCRIPTA, V26, P58

[4]

HAMMOND PR, 1962, J CHEM SOC, P2521

[5]

Kemp BE, 1990, PEPTIDES PROTEIN PHO

[6] ALTERNATIVE STRATEGIES FOR THE FMOC SOLID-PHASE SYNTHESIS OF O-4-PHOSPHO-L-TYROSINE-CONTAINING PEPTIDES [J].

KITAS, EA ;

KNORR, R ;

TRZECIAK, A ;

BANNWARTH, W .

HELVETICA CHIMICA ACTA, 1991, 74 (06) :1314-1328

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