CONTRIBUTION OF RECEPTOR AFFINITY TO ANALGESIC POTENCY

被引:24
作者
TERENIUS, L [1 ]
机构
[1] DEPT MED PHARMACOL UPPSALA,BOX 573,751 23 UPPSALA,SWEDEN
关键词
D O I
10.1111/j.2042-7158.1974.tb09245.x
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:146 / 148
页数:3
相关论文
共 16 条
[1]   DIFFERENCES IN AUTORADIOGRAPHIC LOCALIZATION OF LABELED MORPHINE-LIKE ANALGESICS IN MOUSE [J].
APPELGREN, LE ;
TERENIUS, L .
ACTA PHYSIOLOGICA SCANDINAVICA, 1973, 88 (02) :175-182
[2]  
ASGHAR K, 1970, J PHARMACOL EXP THER, V175, P75
[3]   CENTRAL SITES FOR ANTINOCICEPTIVE ACTION OF MORPHINE AND FENTANYL [J].
HERZ, A ;
ALBUS, K ;
METYS, J ;
SCHUBERT, P ;
TESCHEMACHER, H .
NEUROPHARMACOLOGY, 1970, 9 (06) :539-+
[4]  
HUG CC, 1967, BIOCHEM PHARMACOL, V16, P345
[5]   STRUCTURE-ACTIVITY CORRELATIONS OF MORPHINE-LIKE ANALGETICS BASED ON EFFICIENCIES FOLLOWING INTRAVENOUS AND INTRAVENTRICULAR APPLICATION [J].
KUTTER, E ;
HERZ, A ;
TESCHEMACHER, HJ ;
HESS, R .
JOURNAL OF MEDICINAL CHEMISTRY, 1970, 13 (05) :801-+
[6]   PERSISTENCE OF METHADONE H-3 AND METABOLITE IN RAT-BRAIN AFTER A SINGLE INJECTION AND ITS IMPLICATIONS ON PHARMACOLOGICAL TOLERANCE [J].
MISRA, AL ;
MULE, SJ .
NATURE, 1972, 238 (5360) :155-&
[7]   PROPERTIES OF OPIATE-RECEPTOR BINDING IN RAT-BRAIN [J].
PERT, CB ;
SNYDER, SH .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1973, 70 (08) :2243-2247
[8]   OPIATE RECEPTOR - DEMONSTRATION IN NERVOUS-TISSUE [J].
PERT, CB ;
SNYDER, SH .
SCIENCE, 1973, 179 (4077) :1011-1014
[9]   STEREOSPECIFIC BINDING OF POTENT NARCOTIC ANALGESIC [H-3)ETORPHINE TO RAT-BRAIN HOMOGENATE [J].
SIMON, EJ ;
HILLER, JM ;
EDELMAN, I .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1973, 70 (07) :1947-1949
[10]  
TAKEMORI AE, 1966, J PHARMACOL EXP THER, V154, P586