BIS(HETEROARYL)PIPERAZINE (BHAP) REVERSE-TRANSCRIPTASE INHIBITORS - STRUCTURE-ACTIVITY-RELATIONSHIPS OF NOVEL SUBSTITUTED INDOLE ANALOGS AND THE IDENTIFICATION OF 1-[(5-METHANESULFONAMIDO-1H-INDOL-2-YL)-CARBONYL]-4-[3-[(1-METHYLETHYL)AMINO]-PYRIDINYL]PIPERAZINE MONOMETHANESULFONATE (U-90152S), A 2ND-GENERATION CLINICAL CANDIDATE

被引：135

作者：

ROMERO, DL ^{[1
]}

MORGE, RA ^{[1
]}

GENIN, MJ ^{[1
]}

BILES, C ^{[1
]}

BUSSO, M ^{[1
]}

RESNICK, L ^{[1
]}

ALTHAUS, IW ^{[1
]}

REUSSER, F ^{[1
]}

THOMAS, RC ^{[1
]}

TARPLEY, WG ^{[1
]}

机构：

[1] MT SINAI MED CTR,MIAMI BEACH,FL 33140

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1993年 / 36卷 / 10期

关键词：

D O I：

10.1021/jm00062a027

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：1505 / 1508

页数：4

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