ESTROGEN-RECEPTOR BASED IMAGING AGENTS .1. SYNTHESIS AND RECEPTOR-BINDING AFFINITY OF SOME AROMATIC AND D-RING HALOGENATED ESTROGENS

被引：77

作者：

HEIMAN, DF ^{[1
]}

SENDEROFF, SG ^{[1
]}

KATZENELLENBOGEN, JA ^{[1
]}

NEELEY, RJ ^{[1
]}

机构：

[1] ROGER ADAMS LAB, SCH CHEM SCI, URBANA, IL 61801 USA

来源：

关键词：

D O I：

10.1021/jm00183a007

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：994 / 1002

页数：9

共 71 条

[1] ALBERT S, 1949, J BIOL CHEM, V177, P247
[2] ALLEGRA JC, 1979, CANCER RES, V39, P1447
[3] ALLISON KJ, UNPUBLISHED
[4] ARUNACHALAM T, 1979, J BIOL CHEM, V254, P5900
[5] HETEROCYCLIC FLUORIDES FROM DIAZONIUM FLUOROSILICATES
BEATY, RD
MUSGRAVE, WKR
[J]. JOURNAL OF THE CHEMICAL SOCIETY, 1952, (MAR): : 875 - 878
[6] CHAN RP, 1978, BRIT J PHARMACOL, V63, pP350
[7] COUNSELL RE, 1976, STEROID HORMONE ACTI, P107
[8] DANEK O, 1964, COLLECT CZECH CHEM C, V29, P730
[9] STUDIES IN THE RAT WITH 4-FLUORO-ESTRADIOL-F-18 AND 4-FLUORO-ESTRONE-F-18 AS POTENTIAL PROSTATE SCANNING AGENTS - COMPARISON WITH 2,4-DI-IODO-ESTRADIOL-I-125
EAKINS, MN
PALMER, AJ
WATERS, SL
[J]. INTERNATIONAL JOURNAL OF APPLIED RADIATION AND ISOTOPES, 1979, 30 (11): : 695 - 700
[10] SYNTHESIS OF AROMATIC FLUORIDES THROUGH DIAZOTIZATION IN ANHYDROUS HYDROGEN FLUORIDE
FERM, RL
VANDERWERF, CA
[J]. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1950, 72 (10) : 4809 - 4810