SELECTIVE BLOCKADE OF DOPAMINE D-1 RECEPTOR BY SCH-23390 AFFECTS DOPAMINE AGONIST BINDING TO H-3-SPIPERONE LABELED D-2 RECEPTORS IN RAT STRIATUM

被引:8
作者
ZHANG, X [1 ]
SEGAWA, T [1 ]
机构
[1] HIROSHIMA UNIV,SCH MED,INST PHARMACEUT SCI,DEPT PHARMACOL,KASUMI 1-2-3,MINAMI KU,HIROSHIMA 734,JAPAN
关键词
D O I
10.1254/jjp.50.333
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:333 / 345
页数:13
相关论文
共 40 条
[1]   CHARACTERIZATION OF THE BINDING OF H-3-SCH 23390, A SELECTIVE D-1 RECEPTOR ANTAGONIST LIGAND, IN RAT STRIATUM [J].
BILLARD, W ;
RUPERTO, V ;
CROSBY, G ;
IORIO, LC ;
BARNETT, A .
LIFE SCIENCES, 1984, 35 (18) :1885-1893
[2]   THE D-1 DOPAMINE RECEPTOR ANTAGONIST SCH 23390 ALSO INTERACTS POTENTLY WITH BRAIN-SEROTONIN (5-HT2) RECEPTORS [J].
BISCHOFF, S ;
HEINRICH, M ;
SONNTAG, JM ;
KRAUSS, J .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1986, 129 (03) :367-370
[3]   MECHANISM OF ADENYLATE-CYCLASE ACTIVATION BY CHOLERA TOXIN - INHIBITION OF GTP HYDROLYSIS AT REGULATORY SITE [J].
CASSEL, D ;
SELINGER, Z .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1977, 74 (08) :3307-3311
[4]   THE MAMMALIAN BETA-2-ADRENERGIC RECEPTOR - RECONSTITUTION OF FUNCTIONAL INTERACTIONS BETWEEN PURE RECEPTOR AND PURE STIMULATORY NUCLEOTIDE BINDING-PROTEIN OF THE ADENYLATE-CYCLASE SYSTEM [J].
CERIONE, RA ;
CODINA, J ;
BENOVIC, JL ;
LEFKOWITZ, RJ ;
BIRNBAUMER, L ;
CARON, MG .
BIOCHEMISTRY, 1984, 23 (20) :4519-4525
[5]  
CHATTERJEE TK, 1988, MOL PHARMACOL, V33, P402
[6]   GUANINE-NUCLEOTIDES DISTINGUISH BETWEEN 2 DOPAMINE RECEPTORS [J].
CREESE, I ;
USDIN, T ;
SNYDER, SH .
NATURE, 1979, 278 (5704) :577-578
[7]   H-3-SPIROPERIDOL LABELS SEROTONIN RECEPTORS IN RAT CEREBRAL-CORTEX AND HIPPOCAMPUS [J].
CREESE, I ;
SNYDER, SH .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1978, 49 (02) :201-202
[8]  
CREESE I, 1986, CLIN PHARM, V5, P123
[9]   DOPAMINE RECEPTORS - PHARMACOLOGICAL AND ANATOMICAL EVIDENCES INDICATE THAT 2 DISTINCT DOPAMINE RECEPTOR POPULATIONS ARE PRESENT IN RAT STRIATUM [J].
GARAU, L ;
GOVONI, S ;
STEFANINI, E ;
TRABUCCHI, M ;
SPANO, PF .
LIFE SCIENCES, 1978, 23 (17-1) :1745-1750
[10]   BEHAVIORAL CORRELATIONS OF DOPAMINE RECEPTOR ACTIVATION [J].
GERSHANIK, O ;
HEIKKILA, RE ;
DUVOISIN, RC .
NEUROLOGY, 1983, 33 (11) :1489-1492