STEREOSELECTIVE SYNTHESIS OF A NEW ALDOSE REDUCTASE INHIBITOR - AN EXTENSION OF THE BISLACTIM ETHER METHOD FOR THE SYNTHESIS OF AMINO-ACIDS

被引：4

作者：

GLOMBIK, H

机构：

[1] Hoechst AG

来源：

TETRAHEDRON | 1990年 / 46卷 / 23期

关键词：

D O I：

10.1016/S0040-4020(01)90071-7

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The stereoselective synthesis of the imidazolidinedione (+)-2, an inhibitor of aldose reductase, has been achieved via heterocyclic bislactim ether substitution, acidic cleavage and cyclization with urea. © 1990.

引用

页码：7745 / 7750

页数：6

共 13 条

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