HIGH-THROUGHPUT MICROTITER PLATE-BASED CHROMOGENIC ASSAYS FOR GLYCOSIDASE INHIBITORS

被引:23
作者
WALKER, JM
WINDER, JS
KELLAM, SJ
机构
[1] Division of Biosciences, University of Hertfordshire, Hatfield, AL10 9AB, Herts
关键词
ENZYME INHIBITORS; ALPHA-GLUCOSIDASE; ALPHA-AMYLASE; BETA-GALACTOSIDASE;
D O I
10.1007/BF02916417
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 [生物化学与分子生物学]; 081704 [应用化学];
摘要
Rapid microtiter plate-based colorimetric assays have been developed that allow the screening of large numbers of samples for the presence of inhibitors of alpha-glucosidase, alpha-amylase, and beta-galactosidase. The assays are particularly useful for screening large numbers of microbial culture filtrates.
引用
收藏
页码:141 / 146
页数:6
相关论文
共 18 条
[1]
ISOFLAVONE RHAMUNOSIDES, INHIBITORS OF BETA-GALACTOSIDASE PRODUCED BY ACTINOMYCETES [J].
AOYAGI, T ;
HAZATO, T ;
KUMAGAI, M ;
HAMADA, M ;
TAKEUCHI, T ;
UMEZAWA, H .
JOURNAL OF ANTIBIOTICS, 1975, 28 (12) :1006-1008
[2]
AOYAGI T, 1975, Journal of Antibiotics (Tokyo), V28, P555
[3]
ENZYME INHIBITOR, PANOSIALIN, PRODUCED BY STREPTOMYCES .1. BIOLOGICAL ACTIVITY, ISOLATION AND CHARACTERIZATION OF PANOSIALIN [J].
AOYAGI, T ;
YAGISAWA, M ;
KUMAGAI, M ;
HAMADA, M ;
OKAMI, Y ;
TAKEUCHI, T ;
UMEZAWA, H .
JOURNAL OF ANTIBIOTICS, 1971, 24 (12) :860-&
[4]
THE PRIMARY STRUCTURE OF THE ALPHA-AMYLASE INHIBITOR HOE-467A FROM STREPTOMYCES-TENDAE 4158 - A NEW CLASS OF INHIBITORS [J].
ASCHAUER, H ;
VERTESY, L ;
NESEMANN, G ;
BRAUNITZER, G .
HOPPE-SEYLERS ZEITSCHRIFT FUR PHYSIOLOGISCHE CHEMIE, 1983, 364 (10) :1347-1356
[5]
GLYCOSIDASES IN CANCER AND INVASION [J].
BERNACKI, RJ ;
NIEDBALA, MJ ;
KORYTNYK, W .
CANCER AND METASTASIS REVIEWS, 1985, 4 (01) :81-101
[6]
CANNELL RJP, 1987, J GEN MICROBIOL, V133, P1701
[7]
EFFECT OF CASTANOSPERMINE ON THE STRUCTURE AND SECRETION OF GLYCOPROTEIN ENZYMES IN ASPERGILLUS-FUMIGATUS [J].
ELBEIN, AD ;
MITCHELL, M ;
MOLYNEUX, RJ .
JOURNAL OF BACTERIOLOGY, 1984, 160 (01) :67-75
[8]
INTERFERENCE WITH HIV-INDUCED SYNCYTIUM FORMATION AND VIRAL INFECTIVITY BY INHIBITORS OF TRIMMING GLUCOSIDASE [J].
GRUTERS, RA ;
NEEFJES, JJ ;
TERSMETTE, M ;
DEGOEDE, REY ;
TULP, A ;
HUISMAN, HG ;
MIEDEMA, F ;
PLOEGH, HL .
NATURE, 1987, 330 (6143) :74-77
[9]
INOUYE S, 1968, TETRAHEDRON, V23, P2125
[10]
LAJOLO FM, 1984, NUTR REP INT, V30, P45