ANALOGS OF BETA-LPH61-64 POSSESSING SELECTIVE AGONIST ACTIVITY AT MU-OPIATE RECEPTORS

被引:604
作者
HANDA, BK [1 ]
LANE, AC [1 ]
LORD, JAH [1 ]
MORGAN, BA [1 ]
RANCE, MJ [1 ]
SMITH, CFC [1 ]
机构
[1] RECKITT & COLMAN PHARMACEUT DIV,HULL HU8 7DS,ENGLAND
关键词
D O I
10.1016/0014-2999(81)90364-2
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:531 / 540
页数:10
相关论文
共 23 条
[1]  
BOWER JD, 1980, ENDOGENOUS EXOGENOUS, P29
[2]  
CHANG KJ, 1979, J BIOL CHEM, V254, P2610
[3]  
CHANG KJ, 1979, MOL PHARMACOL, V16, P91
[4]  
GILBERT PE, 1976, J PHARMACOL EXP THER, V198, P66
[5]  
GILLAN MGC, BRIT J PHARMACOL
[6]   MODE OF DEACTIVATION OF ENKEPHALINS BY RAT AND HUMAN-PLASMA AND RAT-BRAIN HOMOGENATES [J].
HAMBROOK, JM ;
MORGAN, BA ;
RANCE, MJ ;
SMITH, CFC .
NATURE, 1976, 262 (5571) :782-783
[7]  
HENDERSHOT LC, 1959, J PHARMACOL EXP THER, V125, P237
[8]   EFFECT OF MORPHINE ON ADRENERGIC TRANSMISSION IN MOUSE VAS-DEFERENS ASSESSMENT OF AGONIST AND ANTAGONIST POTENCIES OF NARCOTIC ANALGESICS [J].
HUGHES, J ;
KOSTERLITZ, HW ;
LESLIE, FM .
BRITISH JOURNAL OF PHARMACOLOGY, 1975, 53 (03) :371-381
[9]   ASSESSMENT IN GUINEA-PIG ILEUM AND MOUSE VAS-DEFERENS OF BENZOMORPHANS WHICH HAVE STRONG ANTINOCICEPTIVE ACTIVITY BUT DO NOT SUBSTITUTE FOR MORPHINE IN DEPENDENT MONKEY [J].
HUTCHINSON, M ;
KOSTERLITZ, HW ;
LESLIE, FM ;
WATERFIELD, AA ;
TERENIUS, L .
BRITISH JOURNAL OF PHARMACOLOGY, 1975, 55 (04) :541-546
[10]  
JANSSEN PAJ, 1963, ARZNEIMITTEL-FORSCH, V13, P502