IS THERE A 2ND EXTERNAL LIDOCAINE BINDING-SITE ON MAMMALIAN CARDIAC-CELLS

被引:74
作者
ALPERT, LA [1 ]
FOZZARD, HA [1 ]
HANCK, DA [1 ]
MAKIELSKI, JC [1 ]
机构
[1] UNIV CHICAGO,MED CTR,CARDIAC ELECTROPHYSIOL LABS,5841 S MARYLAND AVE,BOX 282,CHICAGO,IL 60637
来源
AMERICAN JOURNAL OF PHYSIOLOGY | 1989年 / 257卷 / 01期
关键词
D O I
10.1152/ajpheart.1989.257.1.H79
中图分类号
Q4 [生理学];
学科分类号
071003 ;
摘要
引用
收藏
页码:H79 / H84
页数:6
相关论文
共 23 条
[1]   LIDOCAINE BLOCK OF CARDIAC SODIUM-CHANNELS [J].
BEAN, BP ;
COHEN, CJ ;
TSIEN, RW .
JOURNAL OF GENERAL PHYSIOLOGY, 1983, 81 (05) :613-642
[2]   COOPERATIVITY OF TETRODOTOXIN ACTION IN THE FROG NODE OF RANVIER [J].
BENOIT, E ;
DUBOIS, JM .
PFLUGERS ARCHIV-EUROPEAN JOURNAL OF PHYSIOLOGY, 1985, 405 (03) :237-243
[3]  
BROWN AM, 1981, J PHYSIOL-LONDON, V318, P479
[4]   EVIDENCE FOR A SPECIFIC RECEPTOR-SITE FOR LIDOCAINE, QUINIDINE, AND BUPIVACAINE ASSOCIATED WITH CARDIAC SODIUM-CHANNELS IN GUINEA-PIG VENTRICULAR MYOCARDIUM [J].
CLARKSON, CW ;
HONDEGHEM, LM .
CIRCULATION RESEARCH, 1985, 56 (04) :496-506
[5]  
FRAZIER DT, 1970, J PHARMACOL EXP THER, V171, P45
[6]   THE INFLUENCE OF MOLECULAR-FORM OF LOCAL ANESTHETIC-TYPE ANTI-ARRHYTHMIC AGENTS ON REDUCTION OF THE MAXIMUM UPSTROKE VELOCITY OF CANINE CARDIAC PURKINJE-FIBERS [J].
GINTANT, GA ;
HOFFMAN, BF ;
NAYLOR, RE .
CIRCULATION RESEARCH, 1983, 52 (06) :735-746
[7]  
GINTANT GA, 1987, HDB EXPT PHARMIC, P213
[8]  
GLICKLICH JI, 1978, CIRC RES, V43, P638