PALLADIUM-CATALYZED COUPLING OF URIDINE TRIFLATE WITH ORGANOSTANNANES

被引：35

作者：

CRISP, GT

FLYNN, BL

机构：

[1] Department of Organic Chemistry, University of Adelaide, Adelaide, SA 5001

来源：

TETRAHEDRON LETTERS | 1990年 / 31卷 / 09期

基金：

澳大利亚研究理事会;

关键词：

D O I：

10.1016/S0040-4039(00)88803-6

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

5-Trifluoromethanesulphonyluridine triacetate was readily prepared from 5-hydroxyuridine. This pyrimidine triflate undergoes a palladium-catalysed coupling with vinyl and arylstannanes to give the corresponding 5-substituted uridines. © 1990.

引用

页码：1347 / 1350

页数：4

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