FORMATION OF 6-ACYLINDOLES FROM 1-ACYLINDOLES

被引：23

作者：

NAKATSUKA, S ^{[1
]}

TERANISHI, K ^{[1
]}

GOTO, T ^{[1
]}

机构：

[1] NAGOYA UNIV,SCH AGR,NAGOYA 46401,JAPAN

来源：

TETRAHEDRON LETTERS | 1994年 / 35卷 / 17期

关键词：

D O I：

10.1016/S0040-4039(00)77009-2

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

1-Acylindoles react regioselectively with alpha-halogenoacyl chloride in the presence of aluminum chloride to produce 1-acyl-6-halogenoacylindoles in excellent

引用

页码：2699 / 2700

页数：2

共 6 条

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[3]

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[4] INTRODUCTION OF A HYDROXY GROUP ONTO 5-POSITION AND 6-POSITION OF INDOLE NUCLEUS BY FRIEDEL-CRAFTS ACYLATION AND SUBSEQUENT BAEYER-VILLIGER OXIDATION [J].

NAKATSUKA, S ;

ASANO, O ;

UEDA, K ;

GOTO, T .

HETEROCYCLES, 1987, 26 (06) :1471-1474

[5]

PLANT SGP, 1936, J CHEM SOC, P40

[6]

SUVOROV NN, 1960, J GEN CHEM USSR, V30, P2036

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