CONDENSED HETEROAROMATIC RING-SYSTEMS .24. PALLADIUM-CATALYZED CYCLIZATION OF 2-SUBSTITUTED PHENYLACETYLENES IN THE PRESENCE OF CARBON-MONOXIDE

被引：145

作者：

KONDO, Y ^{[1
]}

SHIGA, F ^{[1
]}

MURATA, N ^{[1
]}

SAKAMOTO, T ^{[1
]}

YAMANAKA, H ^{[1
]}

机构：

[1] TOHOKU UNIV,INST PHARMACEUT,AOBA KU,SENDAI,MIYAGI 98077,JAPAN

来源：

TETRAHEDRON | 1994年 / 50卷 / 41期

关键词：

D O I：

10.1016/S0040-4020(01)89295-4

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The palladium-catalyzed reaction of 2-alkynylanilines and 2-alkynylphenols in the presence of carbon monoxide and methanol under basic conditions gave the sequential cyclization / carbonylation products, methyl 2-substituted indole and benzo[b]-furan-3-carboxylates. Similar reaction of 2-alkynylbenzamides gave 3-alkylidenisoindole derivatives.

引用

页码：11803 / 11812

页数：10

共 12 条

[1] 2-SUBSTITUTED-3-ACYLINDOLES THROUGH THE PALLADIUM-CATALYZED CARBONYLATIVE CYCLIZATION OF 2-ALKYNYLTRIFLUOROACETANILIDES WITH ARYL HALIDES AND VINYL TRIFLATES [J].

ARCADI, A ;

CACCHI, S ;

CARNICELLI, V ;

MARINELLI, F .

TETRAHEDRON, 1994, 50 (02) :437-452

[2]

ARCADI A, 1992, TETRAHEDRON LETT, V33, P3915

[3] PALLADIUM-CATALYZED COUPLING OF ARYL AND VINYL TRIFLATES OR HALIDES WITH 2-ETHYNYLANILINE - AN EFFICIENT ROUTE TO FUNCTIONALIZED 2-SUBSTITUTED INDOLES [J].

ARCADI, A ;

CACCHI, S ;

MARINELLI, F .

TETRAHEDRON LETTERS, 1989, 30 (19) :2581-2584

[4] PALLADIUM CATALYZED REACTION OF 2-ALKYNYLANILINES WITH ALLYL CHLORIDES - FORMATION OF 3-ALLYLINDOLES [J].

IRITANI, K ;

MATSUBARA, S ;

UTIMOTO, K .

TETRAHEDRON LETTERS, 1988, 29 (15) :1799-1802

[5]

KONDO Y, 1989, HETEROCYCLES, V29, P1013

[6] PALLADIUM-CATALYZED SYNTHESIS OF 2-SUBSTITUTED INDOLES [J].

RUDISILL, DE ;

STILLE, JK .

JOURNAL OF ORGANIC CHEMISTRY, 1989, 54 (25) :5856-5866

[7] CONDENSED HETEROAROMATIC RING-SYSTEMS .23. A CONCISE SYNTHESIS OF HIPPADINE [J].

SAKAMOTO, T ;

YASUHARA, A ;

KONDO, Y ;

YAMANAKA, H .

HETEROCYCLES, 1993, 36 (11) :2597-2600

[8]

SAKAMOTO T, 1986, CHEM PHARM BULL, V34, P2754

[9]

SAKAMOTO T, 1992, SYNTHESIS-STUTTGART, P746

[10]

SAKAMOTO T, 1988, CHEM PHARM BULL, V36, P1305

← 1 2 →