PREDICTION OF INTESTINAL 1ST-PASS EFFECT OF PHENACETIN IN THE RAT FROM ENZYME KINETIC DATA - CORRELATION WITH INVIVO DATA USING MUCOSAL BLOOD-FLOW

被引:37
作者
KLIPPERT, P
BORM, P
NOORDHOEK, J
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关键词
D O I
10.1016/0006-2952(82)90068-5
中图分类号
R9 [药学];
学科分类号
1007 ;
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页码:2545 / 2548
页数:4
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共 15 条
  • [1] INTESTINAL MUSCLE AND MUCOSAL BLOOD-FLOW DURING DIRECT SYMPATHETIC STIMULATION
    BOHLEN, HG
    HENRICH, H
    GORE, RW
    JOHNSON, PC
    [J]. AMERICAN JOURNAL OF PHYSIOLOGY, 1978, 235 (01): : H40 - H45
  • [2] INVIVO ASSESSMENT OF EXTRA-HEPATIC CONJUGATIVE METABOLISM IN 1ST PASS EFFECTS USING THE MODEL-COMPOUND PHENOL
    CASSIDY, MK
    HOUSTON, JB
    [J]. JOURNAL OF PHARMACY AND PHARMACOLOGY, 1980, 32 (01) : 57 - 59
  • [3] PHARMACOKINETIC MODEL TO DIFFERENTIATE PREABSORPTIVE, GUT EPITHELIAL, AND HEPATIC 1ST-PASS METABOLISM
    COLBURN, WA
    [J]. JOURNAL OF PHARMACOKINETICS AND BIOPHARMACEUTICS, 1979, 7 (04): : 407 - 415
  • [4] COLBURN WA, 1978, DRUG METAB DISPOS, V6, P193
  • [5] SUBEPITHELIAL CAPILLARY BLOOD-FLOW ESTIMATED FROM BLOOD TO LUMEN FLUX OF BARBITAL IN ILEUM OF RATS
    CSAKY, TZ
    VARGA, F
    [J]. AMERICAN JOURNAL OF PHYSIOLOGY, 1975, 229 (03): : 549 - 552
  • [6] MICROVASCULAR PRESSURES IN RAT INTESTINAL MUSCLE AND MUCOSAL VILLI
    GORE, RW
    BOHLEN, HG
    [J]. AMERICAN JOURNAL OF PHYSIOLOGY, 1977, 233 (06): : H685 - H693
  • [7] GRAFSTROM R, 1979, MED BIOL, V57, P287
  • [8] HULSMANN WC, 1973, METHOD ENZYMOL, V32, P665
  • [9] KLIPPERT PJM, UNPUB J PHARM EXP TH
  • [10] KLIPPERT PJM, UNPUB DRUG METAB DIS