ENANTIOSELECTIVE SYNTHESIS OF ALPHA-AMINO PHOSPHONIC-ACIDS BY AN APPLICATION OF STEREOSELECTIVE OPENING OF HOMOCHIRAL DIOXANE ACETALS WITH TRIETHYL PHOSPHITE

被引：114

作者：

YOKOMATSU, T ^{[1
]}

SHIBUYA, S ^{[1
]}

机构：

[1] TOKYO COLL PHARM,1432-1 HORINOUCHI,HACHIOJI,TOKYO 19203,JAPAN

来源：

TETRAHEDRON-ASYMMETRY | 1992年 / 3卷 / 03期

关键词：

D O I：

10.1016/S0957-4166(00)80280-3

中图分类号：

O61 [无机化学];

学科分类号：

070301 ; 081704 ;

摘要：

Stereoselective opening of homochiral acetals (2a-c) with triethyl phosphite was applied to the enantioselective synthesis of phosphono alcohols (1a-c), which were successfully converted to the alpha-amino phosphonic acid diethyl esters (6a-c).

引用

页码：377 / 378

页数：2

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