EFFECTS OF KETOCONAZOLE ON CHOLESTEROL-SYNTHESIS AND PRECURSOR CONCENTRATIONS IN THE RAT-LIVER

被引:17
作者
STRANDBERG, TE [1 ]
TILVIS, RS [1 ]
MIETTINEN, TA [1 ]
机构
[1] UNIV HELSINKI,DEPT MED 2,SF-00290 HELSINKI 29,FINLAND
关键词
D O I
10.1007/BF02536443
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:1020 / 1024
页数:5
相关论文
共 22 条
[1]   SPECULATIONS ON THE EVOLUTION OF STEROL STRUCTURE AND FUNCTION [J].
BLOCH, KE .
CRC CRITICAL REVIEWS IN BIOCHEMISTRY, 1979, 7 (01) :1-5
[2]  
COOLS W, 1980, ANTIMICROB AGENTS CH, V17, P922
[3]  
ERICKSON SK, 1980, J LIPID RES, V21, P930
[4]  
FOLCH J, 1957, J BIOL CHEM, V226, P497
[5]  
GAYLOR JL, 1968, J BIOL CHEM, V243, P4966
[6]   KETOCONAZOLE - A MAJOR INNOVATION FOR TREATMENT OF FUNGAL DISEASE [J].
GRAYBILL, JR ;
DRUTZ, DJ .
ANNALS OF INTERNAL MEDICINE, 1980, 93 (06) :921-923
[7]   KETOCONAZOLE BLOCKS ADRENAL STEROIDOGENESIS BY INHIBITING CYTOCHROME-P450-DEPENDENT ENZYMES [J].
LOOSE, DS ;
KAN, PB ;
HIRST, MA ;
MARCUS, RA ;
FELDMAN, D .
JOURNAL OF CLINICAL INVESTIGATION, 1983, 71 (05) :1495-1499
[8]  
LOWRY OH, 1951, J BIOL CHEM, V193, P265
[9]  
MIETTINEN TA, 1984, LANCET, V2, P1271
[10]   SERUM SQUALENE AND METHY STEROLS AS INDICATORS OF CHOLESTEROL SYNTHESIS IN VIVO [J].
MIETTINEN, TA .
LIFE SCIENCES PART 1 PHYSIOLOGY AND PHARMACOLOGY AND PART 2 BIOCHEMISTRY GENERAL AND MOLECULAR BIOLOGY, 1969, 8 (14P2) :713-+