USEFUL SYNTHESES OF (3S)-2,3,4,5-TETRAHYDROPYRIDAZINE-3-CARBOXYLIC ACID AND ITS DEHYDROTETRAPEPTIDE DERIVATIVES

被引：21

作者：

NAKAMURA, Y ^{[1
]}

SHIN, C ^{[1
]}

机构：

[1] KANAGAWA UNIV, FAC TECHNOL, ORGAN CHEM LAB, KANAGAWA KU, YOKOHAMA 221, JAPAN

来源：

CHEMISTRY LETTERS | 1991年 / 11期

关键词：

D O I：

10.1246/cl.1991.1953

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

The stereoselective synthesis of (3S)-2,3,4,5-tetrahydropyridazine-3-carboxylic acid (Pya), which is a cyclic alpha-amino acid at center of antrimycins (1), was successful. Moreover, the synthesis of the C-terminal dehydrotetrapeptide of 1 containing Pya residue at N-terminus is described.

引用

页码：1953 / 1956

页数：4

共 5 条

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