CRYSTALLOGRAPHIC STRUCTURAL-ANALYSIS OF PHOSPHORAMIDATES AS INHIBITORS AND TRANSITION-STATE ANALOGS OF THERMOLYSIN

被引：130

作者：

TRONRUD, DE

MONZINGO, AF

MATTHEWS, BW

机构：

[1] UNIV OREGON,INST MOLEC BIOL,EUGENE,OR 97403

[2] UNIV OREGON,DEPT PHYS,EUGENE,OR 97403

[3] UNIV OREGON,DEPT CHEM,EUGENE,OR 97403

来源：

EUROPEAN JOURNAL OF BIOCHEMISTRY | 1986年 / 157卷 / 02期

关键词：

D O I：

10.1111/j.1432-1033.1986.tb09664.x

中图分类号：

Q5 [生物化学]; Q7 [分子生物学];

学科分类号：

071010 ; 081704 ;

摘要：

引用

页码：261 / 268

页数：8

共 34 条

[1] SIMILARITIES IN ACTIVE-CENTER GEOMETRIES OF ZINC-CONTAINING ENZYMES, PROTEASES AND DEHYDROGENASES [J].

ARGOS, P ;

GARAVITO, RM ;

EVENTOFF, W ;

ROSSMANN, MG ;

BRANDEN, CI .

JOURNAL OF MOLECULAR BIOLOGY, 1978, 126 (02) :141-158

[2] PHOSPHONAMIDATES AS TRANSITION-STATE ANALOG INHIBITORS OF THERMOLYSIN [J].

BARTLETT, PA ;

MARLOWE, CK .

BIOCHEMISTRY, 1983, 22 (20) :4618-4624

[3] PROTEIN DATA BANK - COMPUTER-BASED ARCHIVAL FILE FOR MACROMOLECULAR STRUCTURES [J].

BERNSTEIN, FC ;

KOETZLE, TF ;

WILLIAMS, GJB ;

MEYER, EF ;

BRICE, MD ;

RODGERS, JR ;

KENNARD, O ;

SHIMANOUCHI, T ;

TASUMI, M .

JOURNAL OF MOLECULAR BIOLOGY, 1977, 112 (03) :535-542

[4]

BOLOGNESI MC, 1979, J BIOL CHEM, V254, P634

[5] DESIGN OF POTENT COMPETITIVE INHIBITORS OF ANGIOTENSIN-CONVERTING ENZYME - CARBOXYALKANOYL AND MERCAPTOALKANOYL AMINO-ACIDS [J].

CUSHMAN, DW ;

CHEUNG, HS ;

SABO, EF ;

ONDETTI, MA .

BIOCHEMISTRY, 1977, 16 (25) :5484-5491

[6] INHIBITION OF ANGIOTENSIN CONVERTING ENZYME BY PHOSPHORAMIDATES AND POLYPHOSPHATES [J].

GALARDY, RE .

BIOCHEMISTRY, 1982, 21 (23) :5777-5781

[7] INHIBITION OF ANGIOTENSIN CONVERTING ENZYME BY PHOSPHONIC AMIDES AND PHOSPHONIC-ACIDS [J].

GALARDY, RE ;

KONTOYIANNIDOUOSTREM, V ;

KORTYLEWICZ, ZP .

BIOCHEMISTRY, 1983, 22 (08) :1990-1995

[8]

GARDELL SJ, 1986, NATURE LOND

[9] AN INTERACTIVE COMPUTER-GRAPHICS STUDY OF THERMOLYSIN-CATALYZED PEPTIDE CLEAVAGE AND INHIBITION BY N-CARBOXYMETHYL DIPEPTIDES [J].

HANGAUER, DG ;

MONZINGO, AF ;

MATTHEWS, BW .

BIOCHEMISTRY, 1984, 23 (24) :5730-5741

[10] STRUCTURAL-ANALYSIS OF THE INHIBITION OF THERMOLYSIN BY AN ACTIVE-SITE-DIRECTED IRREVERSIBLE INHIBITOR [J].

HOLMES, MA ;

TRONRUD, DE ;

MATTHEWS, BW .

BIOCHEMISTRY, 1983, 22 (01) :236-240

← 1 2 3 4 →