THE 1ST SYNTHESIS OF A MOENOMYCIN-TYPE TRANSGLYCOSYLASE INHIBITOR

被引：16

作者：

LUNING, J

MOLLER, U

MULLER, D

WELZEL, P

MARKUS, A

VANHEIJENOORT, Y

VANHEIJENOORT, J

机构：

[1] RUHR UNIV BOCHUM,FAK CHEM,D-44780 BOCHUM,GERMANY

[2] HOECHST AG,D-65926 FRANKFURT,GERMANY

[3] UNIV PARIS 11,F-91405 ORSAY,FRANCE

来源：

TETRAHEDRON | 1993年 / 49卷 / 46期

关键词：

D O I：

10.1016/S0040-4020(01)81550-7

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Starting from chitobiose octaacetate, D-galacturonic acid derivative 3, and D-glyceric acid derived building block 7, the moenomycin trisaccharide analogue 8c has been synthesized. 8c is an as active transglycosylase inhibitor as moenomycin A.

引用

页码：10587 / 10596

页数：10

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