PARA-[H-3]-META-AZIDOPHENYL ACETIC-ACID, A USEFUL REAGENT FOR THE SYNTHESIS OF RADIOACTIVE PHOTOAFFINITY LIGANDS - SYNTHESIS OF PHOTOAFFINITY-LABELING ECDYSONES

被引：7

作者：

BOEHM, MF

NAKANISHI, K

CHERBAS, P

机构：

[1] COLUMBIA UNIV,DEPT CHEM,NEW YORK,NY 10027

[2] INDIANA UNIV,DEPT BIOL,BLOOMINGTON,IN 47405

来源：

JOURNAL OF THE CHEMICAL SOCIETY-CHEMICAL COMMUNICATIONS | 1991年 / 01期

关键词：

D O I：

10.1039/c39910000052

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

The synthesis of [H-3]-p-azidophenyl acetic acid and its use in the preparation of aryl azido photoaffinity labelled 20-hydroxyecdysone analogues is described.

引用

页码：52 / 53

页数：2

共 19 条

[1]

[Anonymous], INSECT PHYSL

[2]

Bayley H., 1983, PHOTOGENERATED REAGE

[3] THE ECDYSTEROID RECEPTOR [J].

BIDMON, HJ ;

SLITER, TJ .

INVERTEBRATE REPRODUCTION & DEVELOPMENT, 1990, 18 (1-2) :13-27

[4]

Blum M. S., 1985, FUNDAMENTALS INSECT

[5] STRUCTURAL AND FUNCTIONAL-ANALYSIS OF SOME MOLTING HORMONE-RESPONSIVE GENES FROM DROSOPHILA [J].

CHERBAS, L ;

BENES, H ;

BOUROUIS, M ;

BURTIS, K ;

CHAO, A ;

CHERBAS, P ;

CROSBY, M ;

GARFINKEL, M ;

GUILD, G ;

HOGNESS, D ;

JAMI, J ;

JONES, CW ;

KOEHLER, M ;

LEPESANT, JA ;

MARTIN, C ;

MASCHAT, F ;

MATHERS, P ;

MEYEROWITZ, E ;

MOSS, R ;

PICTET, R ;

REBERS, J ;

RICHARDS, G ;

ROUX, J ;

SCHULZ, R ;

SEGRAVES, W ;

THUMMEL, C ;

VIJAYRAGHAVAN, K .

INSECT BIOCHEMISTRY, 1986, 16 (01) :241-248

[6] 26-[I-125]IODOPONASTERONE-A IS A POTENT ECDYSONE AND A SENSITIVE RADIOLIGAND FOR ECDYSONE RECEPTORS [J].

CHERBAS, P ;

CHERBAS, L ;

LEE, SS ;

NAKANISHI, K .

PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1988, 85 (07) :2096-2100

[7]

CHERBAS P, UNPUB

[8] ARYL AZIDES AS PHOTOLABELS - RETENTION OF IODINE DURING PHOTOCHEMICAL RING EXPANSION OF AN IODINATED TYROSINE DERIVATIVE [J].

HENRIKSEN, U ;

BUCHARDT, O .

TETRAHEDRON LETTERS, 1990, 31 (17) :2443-2444

[9]

HIKINO H, 1976, TETRAHEDRON, P3015

[10] PROSTAGLANDIN PHOTOAFFINITY PROBES - SYNTHESIS AND BIOLOGICAL-ACTIVITY OF AZIDE-SUBSTITUTED 16-PHENOXY-PGF2-ALPHA AND 17-PHENYL-PGF2-ALPHA PROSTAGLANDINS [J].

KAWADA, K ;

DOLENCE, EK ;

MORITA, H ;

KOMETANI, T ;

WATT, DS ;

BALAPURE, A ;

FITZ, TA ;

ORLICKY, DJ ;

GERSCHENSON, LE .

JOURNAL OF MEDICINAL CHEMISTRY, 1989, 32 (01) :256-264

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