SHORT CONVERGENT SYNTHESES OF 1,11-EPITHIO AND 1,11-EPOXY STEROIDS

被引：10

作者：

ADAMS, JP

BOWLER, J

COLLINS, MA

JONES, DN

SWALLOW, S

机构：

[1] UNIV SHEFFIELD,DEPT CHEM,SHEFFIELD S3 7HF,S YORKSHIRE,ENGLAND

[2] ICI PLC,MACCLESFIELD SK10 4TG,CHESHIRE,ENGLAND

来源：

TETRAHEDRON LETTERS | 1990年 / 31卷 / 30期

关键词：

D O I：

10.1016/S0040-4039(00)97621-4

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Three component coupling of allyl aryl sulphones with 2-methylcyclopantenone and 2-bromomethylbenzo[b]thiophene or its furan analogue, followed by intramolecular Lewis acid catalysed cyclizations provided short stereoselective syntheses of 1,11-epithio and 1,11-epoxy steroids. © 1990.

引用

页码：4355 / 4358

页数：4

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