PROPOSALS FOR CONFORMATION OF ENKEPHALINS RELATED TO OPIATE MU-PHARMACOPHORE

被引：21

作者：

MAIGRET, B ^{[1
]}

PREMILAT, S ^{[1
]}

FOURNIEZALUSKI, MC ^{[1
]}

ROQUES, BP ^{[1
]}

机构：

[1] UER SCI PHARMACEUT & BIOL,CNRS,EQUIPE RECH 613,DEPT CHIM ORGAN,F-75006 PARIS,FRANCE

来源：

BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS | 1981年 / 99卷 / 01期

关键词：

D O I：

10.1016/0006-291X(81)91741-1

中图分类号：

Q5 [生物化学]; Q7 [分子生物学];

学科分类号：

071010 ; 081704 ;

摘要：

引用

页码：267 / 274

页数：8

共 40 条

[1] STRUCTURAL REQUIREMENTS FOR OPIOID ACTIVITY OF ANALOGS OF ENKEPHALINS
BEDDELL, CR
CLARK, RB
HARDY, GW
LOWE, LA
UBATUBA, FB
VANE, JR
WILKINSON, S
CHANG, KJ
CUATRECASAS, P
MILLER, RJ
[J]. PROCEEDINGS OF THE ROYAL SOCIETY SERIES B-BIOLOGICAL SCIENCES, 1977, 198 (1132): : 249 - 265
[2] BINDING OF FLEXIBLE LIGANDS TO MACROMOLECULES
BURGEN, ASV
ROBERTS, GCK
FEENEY, J
[J]. NATURE, 1975, 253 (5494) : 753 - 755
[3] POSSIBLE ROLE OF DISTINCT MORPHINE AND ENKEPHALIN RECEPTORS IN MEDIATING ACTIONS OF BENZOMORPHAN DRUGS (PUTATIVE-KAPPA AND SIGMA-AGONISTS)
CHANG, KJ
HAZUM, E
CUATRECASAS, P
[J]. PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1980, 77 (08): : 4469 - 4473
[4] OPIATE RECEPTOR-BINDING AFFECTED DIFFERENTIALLY BY OPIATES AND OPIOID PEPTIDES
CHILDERS, SR
CREESE, I
SNOWMAN, AM
SNYDER, SH
[J]. EUROPEAN JOURNAL OF PHARMACOLOGY, 1979, 55 (01) : 11 - 18
[5] OPIATE ACTIVITY OF [DALA2,DELTAZPHE4]-METHIONINE-ENKEPHALINAMIDE
CHIPKIN, RE
STEWART, JM
STAMMER, CH
[J]. BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1979, 87 (03) : 890 - 895
[6] CONFORMATION OF 2,9-DIMETHYL-3'-HYDROXY-5-PHENYL-6,7-BENZOMORPHAN AND ITS RELATION TO OTHER ANALGETICS AND ENKEPHALIN
CLARKE, FH
JAGGI, H
LOVELL, RA
[J]. JOURNAL OF MEDICINAL CHEMISTRY, 1978, 21 (07) : 600 - 606
[7] DIMAIO J, 1979, 6TH P AM PEPT S, P889
[8] OPIATE RECEPTOR - MODEL EXPLAINING STRUCTURE-ACTIVITY-RELATIONSHIPS OF OPIATE AGONISTS AND ANTAGONISTS
FEINBERG, AP
CREESE, I
SNYDER, SH
[J]. PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1976, 73 (11) : 4215 - 4219
[9] ENKEPHALIN RELATED FRAGMENTS - CONFORMATIONAL STUDIES OF TETRAPEPTIDES TYR-GLY-GLY-PHE AND GLY-GLY-PHE-X (X=LEU, MET) BY X-RAY AND H-1 NMR-SPECTROSCOPY
FOURNIEZALUSKI, MC
PRANGE, T
PASCARD, C
ROQUES, BP
[J]. BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1977, 79 (04) : 1199 - 1206
[10] DIFFERENTIATION OF DELTA AND MU OPIATE RECEPTOR LOCALIZATIONS BY LIGHT MICROSCOPIC AUTORADIOGRAPHY
GOODMAN, RR
SNYDER, SH
KUHAR, MJ
YOUNG, WS
[J]. PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1980, 77 (10): : 6239 - 6243

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