NICOTINE ANALOGS - SYNTHESIS OF PYRIDYLAZETIDINES

被引：21

作者：

SECOR, HV

EDWARDS, WB

机构：

[1] Philip Morris Research Center, Richmond

来源：

JOURNAL OF ORGANIC CHEMISTRY | 1979年 / 44卷 / 18期

关键词：

D O I：

10.1021/jo01332a009

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The synthesis of 2-and 3-(3-pyridyl)azetidines (3 and 5) and their IV-methyl derivatives is reported. The key steps involve the preparation of 3-amino-2-(3-pyridyl)-l-propanol (17b) and the reductive detosylation of the N-(4-toluenesulfonyl) derivatives of 3 and 5. © 1979, American Chemical Society. All rights reserved.

引用

页码：3136 / 3140

页数：5

共 35 条

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