FLUORINE-CONTAINING AMINO-ACIDS AND THEIR DERIVATIVES .7. SYNTHESIS AND ANTITUMOR-ACTIVITY OF ALPHA-SUBSTITUTED AND GAMMA-SUBSTITUTED METHOTREXATE ANALOGS

被引：124

作者：

TSUSHIMA, T

KAWADA, K

ISHIHARA, S

UCHIDA, N

SHIRATORI, O

HIGAKI, J

HIRATA, M

机构：

来源：

关键词：

D O I：

10.1016/S0040-4020(01)86044-0

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

引用

页码：5375 / 5387

页数：13

共 76 条

[1] SUICIDE ENZYME INACTIVATORS
ABELES, RH
MAYCOCK, AL
[J]. ACCOUNTS OF CHEMICAL RESEARCH, 1976, 9 (09) : 313 - 319
[2] RECENT ADVANCES IN ASYMMETRIC-SYNTHESIS
APSIMON, JW
SEGUIN, RP
[J]. TETRAHEDRON, 1979, 35 (24) : 2797 - 2842
[3] BERGMANN ED, 1973, SYNTHESIS-STUTTGART, V1, P44
[4] ALKYLATION OF MALONATES OR SCHIFF-BASE ANIONS WITH DICHLOROFLUOROMETHANE AS A ROUTE TO ALPHA-CHLOROFLUOROMETHYL OR ALPHA-FLUOROMETHYL ALPHA-AMINO-ACIDS
BEY, P
DUCEP, JB
SCHIRLIN, D
[J]. TETRAHEDRON LETTERS, 1984, 25 (49) : 5657 - 5660
[5] BEY P, 1977, MED CHEM, V5, P155
[6] BORY S, 1984, INT J PEPT PROT RES, V24, P505
[7] BOSNICH B, 1981, TOP STEREOCHEM, V12, P119
[8] GAMMA-FLUOROGLUTAMIC ACID
BUCHANAN, RL
PATTISON, FL
DEAN, FH
[J]. CANADIAN JOURNAL OF CHEMISTRY-REVUE CANADIENNE DE CHIMIE, 1962, 40 (08): : 1571 - &
[9] INVESTIGATION OF ROLE OF TRYPTOPHAN IN LUTEINIZING HORMONE-RELEASING HORMONE
COY, DH
COY, EJ
HIROTSU, Y
VILCHEZM.JA
SCHALLY, AV
VANNISPE.JW
TESSER, GI
[J]. BIOCHEMISTRY, 1974, 13 (17) : 3550 - 3553
[10] CRAMER SM, 1984, CANCER RES, V44, P1843