EFFECT OF ENKEPHALIN AND ENDORPHIN ANALOGS ON RECEPTORS IN MOUSE VAS-DEFERENS

被引:6
作者
BRITTON, DR
FERTEL, R
COY, DH
KASTIN, AJ
机构
[1] TULANE UNIV, SCH MED, NEW ORLEANS, LA 70112 USA
[2] VET ADM HOSP, NEW ORLEANS, LA 70112 USA
关键词
D O I
10.1016/0006-2952(78)90088-6
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:2275 / 2277
页数:3
相关论文
共 29 条
[1]   ANALGESIA INDUCED INVIVO BY CENTRAL ADMINISTRATION OF ENKEPHALIN IN RAT [J].
BELLUZZI, JD ;
GRANT, N ;
GARSKY, V ;
SARANTAKIS, D ;
WISE, CD ;
STEIN, L .
NATURE, 1976, 260 (5552) :625-626
[2]   ENDORPHINS - PROFOUND BEHAVIORAL-EFFECTS IN RATS SUGGEST NEW ETIOLOGICAL FACTORS IN MENTAL-ILLNESS [J].
BLOOM, F ;
SEGAL, D ;
LING, N ;
GUILLEMIN, R .
SCIENCE, 1976, 194 (4265) :630-632
[3]   BIOSYNTHETIC ORIGIN AND RECEPTOR CONFORMATION OF METHIONINE ENKEPHALIN [J].
BRADBURY, AF ;
SMYTH, DG ;
SNELL, CR .
NATURE, 1976, 260 (5547) :165-166
[4]   COMPARISON OF ANALGESIC PROPERTIES OF LIPOTROPIN C-FRAGMENT AND STABILIZED ENKEPHALINS IN RAT [J].
BRADBURY, AF ;
SMYTH, DG ;
SNELL, CR ;
DEAKIN, JFW ;
WENDLANDT, S .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1977, 74 (02) :748-754
[5]   OPIATE RECEPTOR AFFINITIES AND BEHAVIORAL-EFFECTS OF ENKEPHALIN - STRUCTURE-ACTIVITY RELATIONSHIP OF 10 SYNTHETIC PEPTIDE ANALOGS [J].
CHANG, JK ;
FONG, BTW ;
PERT, A ;
PERT, CB .
LIFE SCIENCES, 1976, 18 (12) :1473-1481
[6]   SYNTHESIS AND OPIOID ACTIVITIES OF STEREOISOMERS AND OTHER D-AMINO-ACID ANALOGS OF METHIONINE-ENKEPHALIN [J].
COY, DH ;
KASTIN, AJ ;
SCHALLY, AV ;
MORIN, O ;
CARON, NG ;
LABRIE, F ;
WALKER, JM ;
FERTEL, R ;
BERNTSON, GG ;
SANDMAN, CA .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1976, 73 (03) :632-638
[7]   COMPARATIVE-STUDY ON ANALGESIC EFFECT OF MET5-ENKEPHALIN AND RELATED LIPOTROPIN FRAGMENTS [J].
GRAF, L ;
SZEKELY, JI ;
RONAI, AZ ;
DUNAIKOVACS, Z ;
BAJUSZ, S .
NATURE, 1976, 263 (5574) :240-241
[8]   MODE OF DEACTIVATION OF ENKEPHALINS BY RAT AND HUMAN-PLASMA AND RAT-BRAIN HOMOGENATES [J].
HAMBROOK, JM ;
MORGAN, BA ;
RANCE, MJ ;
SMITH, CFC .
NATURE, 1976, 262 (5571) :782-783
[9]   NEW EXAMPLE OF A MORPHINE-SENSITIVE NEURO-EFFECTOR JUNCTION - ADRENERGIC TRANSMISSION IN MOUSE VAS-DEFERENS [J].
HENDERSON, G ;
HUGHES, J ;
KOSTERLITZ, HW .
BRITISH JOURNAL OF PHARMACOLOGY, 1972, 46 (04) :764-766
[10]   ENKEPHALINS AND OPIATES - STRUCTURE-ACTIVITY RELATIONS [J].
HORN, AS ;
RODGERS, JR .
JOURNAL OF PHARMACY AND PHARMACOLOGY, 1977, 29 (05) :257-265