SYNTHESIS OF INDOLIZINE-6,9-DIONES ANNELATED TO A THIOPHENE RING

被引：34

作者：

MARCHALIN, S ^{[1
]}

DECROIX, B ^{[1
]}

MOREL, J ^{[1
]}

机构：

[1] UNIV HAVRE, CHIM LAB, F-76600 LE HAVRE, FRANCE

来源：

ACTA CHEMICA SCANDINAVICA | 1993年 / 47卷 / 03期

关键词：

D O I：

10.3891/acta.chem.scand.47-0287

中图分类号：

Q5 [生物化学]; Q7 [分子生物学];

学科分类号：

071010 ; 081704 ;

摘要：

Indolizine-6,9-diones fused to a thiophene ring have been prepared by Friedel-Crafts cyclization of (+/-)-5-oxo-1-(thienylmethyl)prolines. The ketones were converted into oximes, either as syn-anti mixtures or as single isomers. The selectivity of the reaction is discussed.

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页码：287 / 291

页数：5

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