PHYTOGROWTH-INHIBITORY ACTIVITY OF SULFUR-CONTAINING-COMPOUNDS .1. INHIBITORY ACTIVITIES OF THIAZOLIDINE DERIVATIVES ON PLANT-GROWTH

被引:26
作者
INAMORI, Y
MURO, C
TANAKA, R
ADACHI, A
MIYAMOTO, K
TSUJIBO, H
机构
[1] Osaka University of Pharmaceutical Sciences
关键词
(R)-(-)-THIAZOLIDINE-4-CARBOXYLIC ACID; (4R)-(-)-2-THIOXO-4-THIAZOLIDINECARBOXYLIC ACID; 2-THIOXO-4-THIAZOLIDINONE; 4-OXO-2-THIOXOTHIAZOLIDINE-3-ACETIC ACID; THIAZOLIDINE DERIVATIVE; PHYTOGROWTH-INHIBITORY ACTIVITY; BRASSICA-RAPA L; CHLOROPHYLL BIOSYNTHESIS; INHIBITION;
D O I
10.1248/cpb.40.2854
中图分类号
R914 [药物化学];
学科分类号
100701 ;
摘要
(R)-(-)-Thiazolidine-4-carboxylic acid (1, l-thioproline), (4R)-(-)-2-thioxo-4-thiazolidinecarboxylic acid (II), 2-thioxo-4-thiazolidinone (III, rhodanine), 4-oxo-2-thioxothiazolidine-3-acetic acid (IV, rhodanine-3-acetic acid) and thiazolidine (V) showed rather strong inhibitory activity on four kinds of plants examined at the concentration of 3.0 x 10(-4) M. In particular, four compounds except for V strongly inhibited the growth of roots of all the plants examined at the concentration of 1.0 x 10(-3) m. Furthermore, three compounds except for I and V inhibited the germination of the seeds of some plants at the concentration of 1.0 x 10(-3) m. The amount of chlorophyll in the cotyledons of Brassica rapa L. treated with 1.0 x 10(-3) M of I-V was decreased compared to that of the control group. Of the five compounds, III strongly inhibited the chlorophyll biosynthesis of this plant even at the concentration of 3.0 x 10(-4) M.
引用
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页码:2854 / 2856
页数:3
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