BIOLOGY AND MODE OF ACTION OF PURE ANTIOESTROGENS

被引:172
作者
WAKELING, AE
BOWLER, J
机构
关键词
D O I
10.1016/0022-4731(88)90086-6
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
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页码:141 / 147
页数:7
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共 18 条
  • [1] EFFECT OF HYPOPHYSECTOMY AND HORMONE REPLACEMENT ON HORMONE RECEPTOR LEVELS AND THE GROWTH OF 7,12-DIMETHYLBENZ(A)ANTHRACENE-INDUCED MAMMARY-TUMORS IN THE RAT
    ARAFAH, BM
    MANNI, A
    PEARSON, OH
    [J]. ENDOCRINOLOGY, 1980, 107 (05) : 1364 - 1369
  • [2] ANTAGONISM OF ESTROGEN ACTION WITH A NEW BENZOTHIOPHENE DERIVED ANTI-ESTROGEN
    BLACK, LJ
    JONES, CD
    FALCONE, JF
    [J]. LIFE SCIENCES, 1983, 32 (09) : 1031 - 1036
  • [3] BUCOURT R, 1978, J BIOL CHEM, V253, P8221
  • [4] ICI-176,334 - A NOVEL NONSTEROIDAL, PERIPHERALLY SELECTIVE ANTIANDROGEN
    FURR, BJA
    VALCACCIA, B
    CURRY, B
    WOODBURN, JR
    CHESTERSON, G
    TUCKER, H
    [J]. JOURNAL OF ENDOCRINOLOGY, 1987, 113 (03) : R7 - R9
  • [5] ESTRADIOL INDUCTION OF A GLUCOCORTICOID-RESPONSIVE GENE BY A CHIMERIC RECEPTOR
    GREEN, S
    CHAMBON, P
    [J]. NATURE, 1987, 325 (6099) : 75 - 78
  • [6] HAI MTV, 1978, J ENDOCRINOL, V76, P21
  • [7] JORDAN VC, 1984, PHARMACOL REV, V36, P245
  • [8] TAMOXIFEN AS AN ANTI-TUMOUR AGENT - ROLE OF ESTRADIOL AND PROLACTIN
    JORDAN, VC
    KOERNER, S
    [J]. JOURNAL OF ENDOCRINOLOGY, 1976, 68 (02) : 305 - 311
  • [9] DIFFERENTIAL SENSITIVITY OF ESTROGEN TARGET TISSUES - THE ROLE OF THE RECEPTOR
    KELNER, KL
    KIRCHICK, HJ
    PECK, EJ
    [J]. ENDOCRINOLOGY, 1982, 111 (06) : 1986 - 1995
  • [10] DIFFERENTIAL DEPLETION OF CYTOPLASMIC HIGH AFFINITY ESTROGEN RECEPTORS AFTER INVIVO ADMINISTRATION OF ANTIOESTROGENS, CLOMIPHENE, MER-25 AND TAMOXIFEN
    KURL, RN
    MORRIS, ID
    [J]. BRITISH JOURNAL OF PHARMACOLOGY, 1978, 62 (04) : 487 - 493