AN EFFICIENT SYNTHESIS OF CHLORINATED IMIDAZOLES THROUGH TERT-BUTYLDIMETHYLSILYLOXY DERIVATIVES

被引：2

作者：

ESTENNE, G ^{[1
]}

LECLERC, G ^{[1
]}

DODEY, P ^{[1
]}

RENAUT, P ^{[1
]}

机构：

[1] LABS FOURNIER,F-21121 DIJON,FRANCE

来源：

JOURNAL OF HETEROCYCLIC CHEMISTRY | 1994年 / 31卷 / 05期

关键词：

D O I：

10.1002/jhet.5570310503

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The protection of 2-substituted imidazole-5-methanol derivatives by tert-BDMS allowed the chlorination of the heterocycle in position 4 with good yield whereas direct chlorination on the imidazole alcohol was unsuccessful.

引用

页码：1121 / 1123

页数：3

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