THE EFFECT OF ACETAMINOPHEN ON THE DISPOSITION OF FENOLDOPAM - COMPETITION FOR SULFATION

被引:20
作者
ZIEMNIAK, JA [1 ]
ALLISON, N [1 ]
BOPPANA, VK [1 ]
DUBB, J [1 ]
STOTE, R [1 ]
机构
[1] SK&F LABS,DEPT DRUG METAB & CLIN RES & DEV,SWEDELAND,PA 19479
关键词
D O I
10.1038/clpt.1987.28
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:275 / 281
页数:7
相关论文
共 16 条
[1]   RENAL VASODILATORS AND HYPERTENSION [J].
ACKERMAN, DM ;
WEINSTOCK, J ;
WIEBELHAUS, VD ;
BERKOWITZ, B .
DRUG DEVELOPMENT RESEARCH, 1982, 2 (03) :283-297
[2]  
BOPPANA VK, 1984, J CHROMATOGR, V317, P463, DOI 10.1016/S0021-9673(01)91686-3
[3]   USE OF A POSTCOLUMN IMMOBILIZED BETA-GLUCURONIDASE ENZYME REACTOR FOR THE DETERMINATION OF DIASTEREOMERIC GLUCURONIDES OF FENOLDOPAM IN PLASMA AND URINE BY HIGH-PERFORMANCE LIQUID-CHROMATOGRAPHY WITH ELECTROCHEMICAL DETECTION [J].
BOPPANA, VK ;
FONG, KLL ;
ZIEMNIAK, JA ;
LYNN, RK .
JOURNAL OF CHROMATOGRAPHY, 1986, 353 :231-247
[4]  
CALDWELL T, 1978, CONJUGATION REACTION, P477
[5]   THE EFFECT OF ORAL FENOLDOPAM (SKF 82526-J), A PERIPHERAL DOPAMINE RECEPTOR AGONIST, ON BLOOD-PRESSURE AND RENAL-FUNCTION IN NORMAL MAN [J].
HARVEY, JN ;
WORTH, DP ;
BROWN, J ;
LEE, MR .
BRITISH JOURNAL OF CLINICAL PHARMACOLOGY, 1985, 19 (01) :21-27
[6]  
KRIGSHELD KR, 1982, SULFATE METABOLISM S, P59
[7]  
KRIGSHELD KR, 1981, BIOCHEM PHARMACOL, V30, P1973
[8]   DRUG BIOTRANSFORMATION INTERACTIONS IN MAN .3. ACETAMINOPHEN AND SALICYLAMIDE [J].
LEVY, G ;
YAMADA, H .
JOURNAL OF PHARMACEUTICAL SCIENCES, 1971, 60 (02) :215-&
[9]  
LEVY G, 1967, J PHARMACOL EXP THER, V156, P285
[10]   PHARMACOKINETIC CONSEQUENCES AND TOXICOLOGIC IMPLICATIONS OF ENDOGENOUS COSUBSTRATE DEPLETION [J].
LEVY, G ;
GALINSKY, RE ;
LIN, JH .
DRUG METABOLISM REVIEWS, 1982, 13 (06) :1009-1020