A FACILE, HIGH-YIELDING METHOD FOR THE CONVERSION OF HALIDES TO MERCAPTANS

被引：18

作者：

BIENIARZ, C

CORNWELL, MJ

机构：

[1] Diagnostics Division, Department of Immunochemistry Abbott Laboratories, Abbott Park

来源：

TETRAHEDRON LETTERS | 1993年 / 34卷 / 06期

关键词：

D O I：

10.1016/S0040-4039(00)77459-4

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

An efficient, high-yield, one-pot preparation of alkyl and activated aryl mercaptans is presented. The method relies on sodium thiophosphate displacement of the halide, followed by mild hydrolysis of the intermediate phosphorothioate.

引用

页码：939 / 942

页数：4

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