ASYMMETRIC-SYNTHESIS OF CALYCULIN-A .3. ASSEMBLAGE OF THE CALYCULIN SKELETON AND THE INTRODUCTION OF A NEW PHOSPHATE MONOESTER SYNTHESIS

被引：42

作者：

EVANS, DA

GAGE, JR

LEIGHTON, JL

机构：

[1] Department of Chemistry, Harvard University, Cambridge

来源：

JOURNAL OF ORGANIC CHEMISTRY | 1992年 / 57卷 / 07期

关键词：

D O I：

10.1021/jo00033a011

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The synthesis of a fully protected analogue of calyculin A has been accomplished using a Wittig reaction to couple two fragments comprising the C1-C25 and C26-C37 portions of calyculin A. Associated model studies on the incorporation of the C17 phosphate monoester moiety are also described.

引用

页码：1964 / 1966

页数：3

共 11 条

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