INVIVO LABELING OF CENTRAL BENZODIAZEPINE RECEPTORS WITH THE PARTIAL INVERSE AGONIST [H-3]RO 15-4513

被引:15
作者
SADZOT, B
FROST, JJ
WAGNER, HN
机构
[1] JOHNS HOPKINS UNIV,SCH MED,DEPT RADIOL,DIV NUCL MED,BALTIMORE,MD 21205
[2] JOHNS HOPKINS UNIV,SCH MED,DEPT NEUROSCI,BALTIMORE,MD 21205
关键词
D O I
10.1016/0006-8993(89)90094-2
中图分类号
Q189 [神经科学];
学科分类号
071006 ;
摘要
引用
收藏
页码:128 / 135
页数:8
相关论文
共 35 条
[1]   BINDING OF [H-3] RO 5-4864 AND [H-3] PK 11195 TO CEREBRAL-CORTEX AND PERIPHERAL-TISSUES OF VARIOUS SPECIES - SPECIES-DIFFERENCES AND HETEROGENEITY IN PERIPHERAL BENZODIAZEPINE BINDING-SITES [J].
AWAD, M ;
GAVISH, M .
JOURNAL OF NEUROCHEMISTRY, 1987, 49 (05) :1407-1414
[2]  
BONETTI EP, 1984, NEUROSCI LETT S, V18, pS30
[3]  
Bonetti EP, 1985, BRIT J PHARMACOL, V86, P463
[4]   BINDING OF [DMCM-H-3, A CONVULSIVE BENZODIAZEPINE LIGAND, TO RAT-BRAIN MEMBRANES - PRELIMINARY STUDIES [J].
BRAESTRUP, C ;
NIELSEN, M ;
HONORE, T .
JOURNAL OF NEUROCHEMISTRY, 1983, 41 (02) :454-465
[5]   [H-3]-LABELED PROPYL BETA-CARBOLINE-3-CARBOXYLATE AS A SELECTIVE RADIOLIGAND FOR THE BZ1 BENZODIAZEPINE RECEPTOR SUBCLASS [J].
BRAESTRUP, C ;
NIELSEN, M .
JOURNAL OF NEUROCHEMISTRY, 1981, 37 (02) :333-341
[6]   THE KINETICS AND DISPLACEMENT OF [FLUNITRAZEPAM-C-11 IN THE BRAIN OF THE LIVING BABOON [J].
COMAR, D ;
MAZIERE, M ;
CEPEDA, C ;
GODOT, JM ;
MENINI, C ;
NAQUET, R .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1981, 75 (01) :21-26
[7]   PROTECTION AGAINST ETHANOL MORTALITY IN RATS BY THE IMIDAZOBENZODIAZEPINE RO 15-4513 [J].
FADDA, F ;
MOSCA, E ;
COLOMBO, G ;
GESSA, GL .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1987, 136 (02) :265-266
[8]  
FROST JJ, 1987, LIFE SCI, V40, P987
[9]   KINETICS OF BINDING TO OPIATE RECEPTORS INVIVO PREDICTED FROM INVITRO PARAMETERS [J].
FROST, JJ ;
WAGNER, HN .
BRAIN RESEARCH, 1984, 305 (01) :1-11
[10]  
FROST JJ, 1986, EUR J PHARMACOL, V122, P381