2-ARYLINDENES AND 2-ARYLINDENONES - SYNTHESIS OF PROBES TO STUDY THE BINDING ORIENTATION OF UNSYMMETRICAL NONSTEROIDAL LIGANDS TO THE ESTROGEN-RECEPTOR

被引：55

作者：

ANSTEAD, GM ^{[1
]}

ENSIGN, JL ^{[1
]}

PETERSON, CS ^{[1
]}

KATZENELLENBOGEN, JA ^{[1
]}

机构：

[1] UNIV ILLINOIS,DEPT CHEM,1209 W CALIF ST,URBANA,IL 61801

来源：

JOURNAL OF ORGANIC CHEMISTRY | 1989年 / 54卷 / 07期

关键词：

D O I：

10.1021/jo00268a003

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

引用

页码：1485 / 1491

页数：7

共 30 条

[1]

[Anonymous], 1963, FREIDEL CRAFTS REL

[2] FLUORESCENCE PROPERTIES OF 2,3-DIARYLINDENES [J].

ANSTEAD, GM ;

KATZENELLENBOGEN, JA .

JOURNAL OF PHYSICAL CHEMISTRY, 1988, 92 (22) :6249-6258

[3] OPTIMIZING OF 2,3-DIARYLINDENES AS FLUORESCENT ESTROGENS - VARIATION OF THE ACCEPTOR GROUP, ORTHO SUBSTITUTION OF THE 2-RING, AND C-1 METHYLATION [J].

ANSTEAD, GM ;

KATZENELLENBOGEN, JA .

JOURNAL OF MEDICINAL CHEMISTRY, 1988, 31 (09) :1754-1761

[4] 2,3-DIARYLINDENES AND 2,3-DIARYLINDENONES - SYNTHESIS, MOLECULAR-STRUCTURE, PHOTOCHEMISTRY, ESTROGEN-RECEPTOR BINDING-AFFINITY, AND COMPARISONS WITH RELATED TRIARYLETHYLENES [J].

ANSTEAD, GM ;

ALTENBACH, RJ ;

WILSON, SR ;

KATZENELLENBOGEN, JA .

JOURNAL OF MEDICINAL CHEMISTRY, 1988, 31 (07) :1316-1326

[5]

ANSTEAD GM, UNPUB J MED CHEM

[6]

ANSTEAD GM, 1987, 194TH NAT M AM CHEM

[7]

ANSTEAD GM, UNPUB PHOTOCHEM PHOT

[8] KINETICS OF IONIZATION OF 1,3-INDANDIONE IN ME2SO WATER MIXTURES - SOLVENT EFFECT ON INTRINSIC RATES AND BRONSTED COEFFICIENTS [J].

BERNASCONI, CF ;

PASCHALIS, P .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1986, 108 (11) :2969-2977

[9] ACIDITIES OF INDENE AND PHENYLINDENES, DIPHENYLINDENES, AND TRIPHENYLINDENES [J].

BORDWELL, FG ;

DRUCKER, GE .

JOURNAL OF ORGANIC CHEMISTRY, 1980, 45 (16) :3325-3328

[10]

BROOME J, 1960, J AM CHEM SOC, V82, P1406

← 1 2 3 →