CONVENIENT PREPARATION OF ALPHA-TERT-BUTYL N-BLOCKED GLUTAMATES THROUGH GAMMA-ALLYL ESTER PROTECTION

被引：5

作者：

BAVETSIAS, V

BISSET, GMF

JARMAN, M

机构：

[1] CRC Centre for Cancer Therapeutics at the Institute of Cancer Research, Chemistry Department, CRC Laboratories, Sutton, Surrey SM2 5NG

来源：

SYNTHETIC COMMUNICATIONS | 1995年 / 25卷 / 07期

关键词：

D O I：

10.1080/00397919508012656

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Utilisation of gamma-allyl ester protection of glutamates provides a convenient route to the synthesis of Z-Glu-OBu(t), Tr-Glu-OBu(t) and (Boc)(2)-Glu-OBu(t).

引用

页码：947 / 958

页数：12

共 7 条

[1] SYNTHESIS OF NONPROTEINOGENIC AMINO-ACIDS .2. PREPARATION OF A SYNTHETIC EQUIVALENT OF THE GAMMA-ANION SYNTHON FOR ASYMMETRIC AMINO-ACID SYNTHESIS
BALDWIN, JE
NORTH, M
FLINN, A
MOLONEY, MG
[J]. TETRAHEDRON, 1989, 45 (05) : 1453 - 1464
[2] SYNTHESIS OF NONPROTEINOGENIC AMINO-ACIDS .3. CONVERSION OF GLUTAMIC-ACID INTO GAMMA,DELTA-UNSATURATED ALPHA-AMINO-ACIDS
BALDWIN, JE
NORTH, M
FLINN, A
MOLONEY, MG
[J]. TETRAHEDRON, 1989, 45 (05) : 1465 - 1474
[3] CHLOROTRIMETHYLSILANE MEDIATED FORMATION OF OMEGA-ALLYL ESTERS OF ASPARTIC AND GLUTAMIC ACIDS
BELSHAW, PJ
MZENGEZA, S
LAJOIE, GA
[J]. SYNTHETIC COMMUNICATIONS, 1990, 20 (20) : 3157 - 3160
[4] PREPARATION OF SEMIALDEHYDE DERIVATIVES OF ASPARTIC AND GLUTAMIC-ACID VIA THE ROSENMUND REDUCTION
BOLD, G
STEINER, H
MOESCH, L
WALLISER, B
[J]. HELVETICA CHIMICA ACTA, 1990, 73 (02) : 405 - 410
[5] A NEW SYNTHESIS OF COPRINE AND O-ETHYLCOPRINE
KIENZLER, T
STRAZEWSKI, P
TAMM, C
[J]. HELVETICA CHIMICA ACTA, 1992, 75 (04) : 1078 - 1084
[6] IMPROVED SYNTHESIS OF SOME ALPHA-ESTERS OF N-PROTECTED L-GLUTAMIC ACID
PAWELCZAK, K
KRZYZANOWSKI, L
RZESZOTARSKA, B
[J]. ORGANIC PREPARATIONS AND PROCEDURES INTERNATIONAL, 1985, 17 (06) : 416 - 419
[7] Rosowsky A, 1989, Prog Med Chem, V26, P1, DOI 10.1016/S0079-6468(08)70241-8

← 1 →