A NOVEL PYRAZOLOQUINOLINE THAT INTERACTS WITH BRAIN BENZODIAZEPINE RECEPTORS - CHARACTERIZATION OF SOME INVITRO AND INVIVO PROPERTIES OF CGS-9896

被引:46
作者
GEE, KW
YAMAMURA, HI
机构
[1] UNIV ARIZONA,ARIZONA HLTH SCI CTR,DEPT BIOCHEM,TUCSON,AZ 85724
[2] UNIV ARIZONA,ARIZONA HLTH SCI CTR,DEPT PSYCHIAT,TUCSON,AZ 85724
[3] UNIV ARIZONA,ARIZONA RES LABS,TUCSON,AZ 85724
关键词
D O I
10.1016/0024-3205(82)90251-X
中图分类号
R-3 [医学研究方法]; R3 [基础医学];
学科分类号
1001 ;
摘要
引用
收藏
页码:2245 / 2252
页数:8
相关论文
共 20 条
  • [1] PHARMACOLOGICAL CHARACTERIZATION OF BENZODIAZEPINE RECEPTORS IN BRAIN
    BRAESTRUP, C
    SQUIRES, RF
    [J]. EUROPEAN JOURNAL OF PHARMACOLOGY, 1978, 48 (03) : 263 - 270
  • [2] URINARY AND BRAIN BETA-CARBOLINE-3-CARBOXYLATES AS POTENT INHIBITORS OF BRAIN BENZODIAZEPINE RECEPTORS
    BRAESTRUP, C
    NIELSEN, M
    OLSEN, CE
    [J]. PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1980, 77 (04): : 2288 - 2292
  • [3] IS THE BENZODIAZEPINE RECEPTOR COUPLED TO A CHLORIDE ANION CHANNEL
    COSTA, T
    RODBARD, D
    PERT, CB
    [J]. NATURE, 1979, 277 (5694) : 315 - 317
  • [4] CGS-8216 - RECEPTOR-BINDING CHARACTERISTICS OF A POTENT BENZODIAZEPINE ANTAGONIST
    CZERNIK, AJ
    PETRACK, B
    KALINSKY, HJ
    PSYCHOYOS, S
    CASH, WD
    TSAI, C
    RINEHART, RK
    GRANAT, FR
    LOVELL, RA
    BRUNDISH, DE
    WADE, R
    [J]. LIFE SCIENCES, 1982, 30 (04) : 363 - 372
  • [5] EHLERT FJ, 1981, LIFE SCI, V29, P235, DOI 10.1016/0024-3205(81)90239-3
  • [6] EHLERT FJ, 1982, EUR J PHARM
  • [7] Greenblatt D. J., 1974, BENZODIAZEPINES CLIN
  • [8] Lippa A., 1979, ANXIOLYTICS, P41
  • [9] BENZODIAZEPINE RECEPTORS - CELLULAR AND BEHAVIORAL-CHARACTERISTICS
    LIPPA, AS
    CRITCHETT, D
    SANO, MC
    KLEPNER, CA
    GREENBLATT, EN
    COUPET, J
    BEER, B
    [J]. PHARMACOLOGY BIOCHEMISTRY AND BEHAVIOR, 1979, 10 (05) : 831 - 843
  • [10] THE ROLE OF GABA IN MEDIATING THE ANTICONVULSANT PROPERTIES OF BENZODIAZEPINES
    LIPPA, AS
    KLEPNER, CA
    BENSON, DI
    CRITCHETT, DJ
    SANO, MC
    BEER, B
    [J]. BRAIN RESEARCH BULLETIN, 1980, 5 : 861 - 865