STRUCTURE-ACTIVITY RELATIONSHIP, SELECTIVITY AND MODE OF INHIBITION OF TERMINAL DEOXYRIBONUCLEOTIDYLTRANSFERASE BY STREPTOLYDIGIN ANALOGS

被引:12
作者
DICIOCCIO, RA
SRIVASTAVA, BIS
RINEHART, KL
LEE, VJ
BRANFMAN, AR
LI, LH
机构
[1] NEW YORK STATE DEPT HLTH,ROSWELL PK MEM INST,GRACE CANC DRUG CTR,BUFFALO,NY 14263
[2] UPJOHN CO,CANC RES,KALAMAZOO,MI 49001
[3] UNIV ILLINOIS,ROGER ADAMS LAB,URBANA,IL 61801
关键词
D O I
10.1016/0006-2952(80)90484-0
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:2001 / 2008
页数:8
相关论文
共 18 条
[1]  
ALBERTS P, 1976, J BIOL CHEM, V251, P1543
[2]  
BRADFORD MM, 1976, ANAL BIOCHEM, V72, P248, DOI 10.1016/0003-2697(76)90527-3
[3]   COMPARISON OF EFFECTS OF L-DOPA, AMPHETAMINE AND APOMORPHINE ON FIRING RATE OF RAT DOPAMINERGIC NEURONS [J].
BUNNEY, BS ;
AGHAJANIAN, GK ;
ROTH, RH .
NATURE-NEW BIOLOGY, 1973, 245 (143) :123-125
[4]  
CLEMENTCORMIER Y, 1978, RES COMMUN CHEM PATH, V22, P15
[5]  
CLEMENTCORMIER Y, 1978, LIFE SCI, V23, P539
[6]   MULTIPLE DOPAMINE BINDING-SITES - SUBCELLULAR-LOCALIZATION AND BIOCHEMICAL CHARACTERIZATION [J].
CLEMENTCORMIER, YC ;
GEORGE, RJ .
JOURNAL OF NEUROCHEMISTRY, 1979, 32 (03) :1061-1069
[7]   SOLUBILIZATION AND CHARACTERIZATION OF [H-3]SPIROPERIDOL BINDING-SITES FROM SUBCELLULAR-FRACTIONS OF THE CALF STRIATUM [J].
CLEMENTCORMIER, YC ;
KENDRICK, PE .
BIOCHEMICAL PHARMACOLOGY, 1980, 29 (06) :897-903
[8]   DOPAMINE RECEPTORS - SELECTIVE AGONISTS AND ANTAGONISTS OF FUNCTIONALLY DISTINCT TYPES WITHIN FELINE BRAIN [J].
COOLS, AR ;
STRUYKERBOUDIER, HAJ ;
VANROSSUM, JM .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1976, 37 (02) :283-293
[9]   DOPAMINE RECEPTOR-BINDING OF ADTN-H-3 (2-AMINO-6,7-DIHYDROXY-1,2,3,4-TETRAHYDRONAPHTHALENE) REGULATED BY GUANYL NUCLEOTIDES [J].
CREESE, I ;
SNYDER, SH .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1978, 50 (04) :459-461
[10]   H-3-SPIROPERIDOL LABELS DOPAMINE RECEPTORS IN PITUITARY AND BRAIN [J].
CREESE, I ;
SCHNEIDER, R ;
SNYDER, SH .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1977, 46 (04) :377-381