KELATORPHAN, A POTENT ENKEPHALINASES INHIBITOR, PRESENTS OPPOSITE PROPERTIES WHEN INJECTED INTRACEREBROVENTRICULARLY OR INTO THE NUCLEUS ACCUMBENS ON INTRACRANIAL SELF-STIMULATION

被引:10
作者
HEIDBREDER, C
ROQUES, B
VANDERHAEGHEN, JJ
DEWITTE, P
机构
[1] UNIV DESCARTES,CHIM ORGAN LAB,PARIS,FRANCE
[2] UNIV LIBRE BRUXELLES,NEUROPEPTIDES LAB,B-1000 BRUSSELS,BELGIUM
关键词
D O I
10.1016/0197-0186(88)90173-8
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:347 / 350
页数:4
相关论文
共 23 条
[1]   BIDENTATE PEPTIDES - HIGHLY POTENT NEW INHIBITORS OF ENKEPHALIN DEGRADING ENZYMES [J].
BOUBOUTOU, R ;
WAKSMAN, G ;
DEVIN, J ;
FOURNIEZALUSKI, MC ;
ROQUES, BP .
LIFE SCIENCES, 1984, 35 (09) :1023-1030
[2]   MORPHINE AND DELTA-OPIATE AGONISTS LOCALLY STIMULATE INVIVO DOPAMINE RELEASE IN CAT CAUDATE-NUCLEUS [J].
CHESSELET, MF ;
CHERAMY, A ;
REISINE, TD ;
GLOWINSKI, J .
NATURE, 1981, 291 (5813) :320-322
[3]   INDUCTION OF CATALEPSY AND HYPERACTIVITY BY MORPHINE ADMINISTERED DIRECTLY INTO NUCLEUS ACCUMBENS OF RATS [J].
COSTALL, B ;
FORTUNE, DH ;
NAYLOR, RJ .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1978, 49 (01) :49-64
[4]   OPPOSITE EFFECTS OF CHOLECYSTOKININ OCTAPEPTIDE (CCK-8) AND TETRAPEPTIDE (CCK-4) AFTER INJECTION INTO THE CAUDAL PART OF THE NUCLEUS-ACCUMBENS OR INTO ITS ROSTRAL PART AND THE CEREBRAL-VENTRICLES [J].
DEWITTE, P ;
HEIDBREDER, C ;
ROQUES, B ;
VANDERHAEGHEN, JJ .
NEUROCHEMISTRY INTERNATIONAL, 1987, 10 (04) :473-479
[5]   BEHAVIORAL DISSOCIATION OF ENCEPHALINERGIC SYSTEMS OF NUCLEUS ACCUMBENS AND NUCLEUS CAUDATUS [J].
DILL, RE ;
COSTA, E .
NEUROPHARMACOLOGY, 1977, 16 (05) :323-326
[7]   CHOLECYSTOKININ PEPTIDES PRODUCE MARKED REDUCTION OF DOPAMINE TURNOVER IN DISCRETE AREAS IN THE RAT-BRAIN FOLLOWING INTRAVENTRICULAR-INJECTION [J].
FUXE, K ;
ANDERSSON, K ;
LOCATELLI, V ;
AGNATI, LF ;
HOKFELT, T ;
SKIRBOLL, L ;
MUTT, V .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1980, 67 (2-3) :329-331
[8]  
HOEBEL BG, 1982, NEURAL BASIS FEEDING
[9]   DETERMINATION OF METHIONINE ENKEPHALIN IN DISCRETE REGIONS OF RAT-BRAIN [J].
HONG, JS ;
YANG, HYT ;
FRATTA, W ;
COSTA, E .
BRAIN RESEARCH, 1977, 134 (02) :383-386
[10]  
IVERSEN SD, 1983, NEUROBIOLOGY OPIATE, P439