SYNTHESIS OF A PHOTOAFFINITY ANALOG OF TAXOL AS AN APPROACH TO IDENTIFY THE TAXOL BINDING-SITE ON MICROTUBULES

被引：27

作者：

CARBONI, JM

FARINA, V

RAO, S

HAUCK, SI

HORWITZ, SB

RINGEL, I

机构：

[1] BRISTOL MYERS SQUIBB RES INST,DEPT EXPTL THERAPEUT,WALLINGFORD,CT 06492

[2] BRISTOL MYERS SQUIBB RES INST,ANTITUMOR CHEM,WALLINGFORD,CT 06492

[3] YESHIVA UNIV ALBERT EINSTEIN COLL MED,DEPT MOLEC PHARMACOL,BRONX,NY 10461

[4] HEBREW UNIV JERUSALEM,HADASSAH MED SCH,DEPT PHARMACOL,IL-91010 JERUSALEM,ISRAEL

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1993年 / 36卷 / 04期

关键词：

D O I：

10.1021/jm00056a013

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

[No abstract available]

引用

页码：513 / 515

页数：3

共 18 条

[1] SYNTHESIS OF A PHOTOREACTIVE TAXOL SIDE-CHAIN
CHATTERJEE, A
WILLIAMSON, JS
ZJAWIONY, JK
PETERSON, JR
[J]. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 1992, 2 (01) : 91 - 94
[2] SELECTIVE CLEAVAGE OF THE ALLYL AND ALLYLOXCARBONYL GROUPS THROUGH PALLADIUM-CATALYZED HYDROSTANNOLYSIS WITH TRIBUTYLTIN HYDRIDE - APPLICATION TO THE SELECTIVE PROTECTION-DEPROTECTION OF AMINO-ACID DERIVATIVES AND IN PEPTIDE-SYNTHESIS
DANGLES, O
GUIBE, F
BALAVOINE, G
LAVIELLE, S
MARQUET, A
[J]. JOURNAL OF ORGANIC CHEMISTRY, 1987, 52 (22) : 4984 - 4993
[3] LARGE RATE ACCELERATIONS IN THE STILLE REACTION WITH TRI-2-FURYLPHOSPHINE AND TRIPHENYLARSINE AS PALLADIUM LIGANDS - MECHANISTIC AND SYNTHETIC IMPLICATIONS
FARINA, V
KRISHNAN, B
[J]. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1991, 113 (25) : 9585 - 9595
[4] TAXOL PHOTOAFFINITY LABEL - 7-(PARA-AZIDOBENZOYL)TAXOL SYNTHESIS AND BIOLOGICAL EVALUATION
GEORG, GI
HARRIMAN, GCB
HIMES, RH
MEJILLANO, MR
[J]. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 1992, 2 (07) : 735 - 738
[5] THE CHEMISTRY OF TAXOL, A CLINICALLY USEFUL ANTICANCER AGENT
KINGSTON, DGI
SAMARANAYAKE, G
IVEY, CA
[J]. JOURNAL OF NATURAL PRODUCTS, 1990, 53 (01): : 1 - 12
[6] THE CHEMISTRY OF TAXOL
KINGSTON, DGI
[J]. PHARMACOLOGY & THERAPEUTICS, 1991, 52 (01) : 1 - 34
[7] PHOTOGENERATED REAGENTS FOR BIOLOGICAL RECEPTOR-SITE LABELING
KNOWLES, JR
[J]. ACCOUNTS OF CHEMICAL RESEARCH, 1972, 5 (04) : 155 - &
[8] PREPARATION AND BIOLOGICAL-ACTIVITY OF TAXOL ACETATES
MELLADO, W
MAGRI, NF
KINGSTON, DGI
GARCIAARENAS, R
ORR, GA
HORWITZ, SB
[J]. BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1984, 124 (02) : 329 - 336
[9] STRUCTURE-ACTIVITY STUDY OF CYTO-TOXICITY AND MICROTUBULE ASSEMBLY INVITRO BY TAXOL AND RELATED TAXANES
PARNESS, J
KINGSTON, DGI
POWELL, RG
HARRACKSINGH, C
HORWITZ, SB
[J]. BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1982, 105 (03) : 1082 - 1089
[10] TAXOL BINDS TO POLYMERIZED TUBULIN INVITRO
PARNESS, J
HORWITZ, SB
[J]. JOURNAL OF CELL BIOLOGY, 1981, 91 (02) : 479 - 487

← 1 2 →