PROSTAGLANDIN-F2-ALPHA PHOTOAFFINITY PROBES - 18-PHENOXY-19,20-BISNORPROSTANOIDS BEARING PERFLUORINATED ARYL AZIDES

被引：6

作者：

GOLINSKI, M ^{[1
]}

HEINE, M ^{[1
]}

WATT, DS ^{[1
]}

机构：

[1] UNIV KENTUCKY,DEPT CHEM,LEXINGTON,KY 40506

来源：

TETRAHEDRON LETTERS | 1991年 / 32卷 / 12期

关键词：

D O I：

10.1016/S0040-4039(00)74270-5

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The synthesis of a potential prostaglandin F2-alpha photoaffinity probe involved the preparation of an 18-phenoxy-19,20-bisnorprostanoid in which the phenoxy group possessed an iodine substituent and a perfluorinated aryl azide.

引用

页码：1553 / 1556

页数：4

共 28 条

[1] CATECHOL BORON HALIDES - MILD AND SELECTIVE REAGENTS FOR CLEAVAGE OF COMMON PROTECTING GROUPS [J].

BOECKMAN, RK ;

POTENZA, JC .

TETRAHEDRON LETTERS, 1985, 26 (11) :1411-1414

[2]

CAI SX, 1989, TETRAHEDRON LETT, V30, P5409

[3] TOTAL SYNTHESIS OF MAYTANSINE [J].

COREY, EJ ;

WEIGEL, LO ;

CHAMBERLIN, AR ;

CHO, H ;

HUA, DH .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1980, 102 (21) :6613-6615

[4] STEREO-CONTROLLED SYNTHESIS OF PROSTAGLANDINS F2ALPHA AND E2 (DL) [J].

COREY, EJ ;

WEINSHENKER, NM ;

SCHAAF, TK ;

HUBER, W .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1969, 91 (20) :5675-+

[5] PROTECTION OF HYDROXYL GROUPS AS TERT-BUTYLDIMETHYLSILYL DERIVATIVES [J].

COREY, EJ ;

VENKATESWARLU, A .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1972, 94 (17) :6190-+

[6]

COREY EJ, 1976, TETRAHEDRON LETT, V17, P809

[7] QUANTITATIVE DEALKYLATION OF ALKYL ETHERS VIA TREATMENT WITH TRIMETHYLSILYL IODIDE - NEW METHOD FOR ETHER HYDROLYSIS [J].

JUNG, ME ;

LYSTER, MA .

JOURNAL OF ORGANIC CHEMISTRY, 1977, 42 (23) :3761-3764

[8] PROSTAGLANDIN PHOTOAFFINITY PROBES - SYNTHESIS AND BIOLOGICAL-ACTIVITY OF AZIDE-SUBSTITUTED 16-PHENOXY-PGF2-ALPHA AND 17-PHENYL-PGF2-ALPHA PROSTAGLANDINS [J].

KAWADA, K ;

DOLENCE, EK ;

MORITA, H ;

KOMETANI, T ;

WATT, DS ;

BALAPURE, A ;

FITZ, TA ;

ORLICKY, DJ ;

GERSCHENSON, LE .

JOURNAL OF MEDICINAL CHEMISTRY, 1989, 32 (01) :256-264

[9] FUNCTIONALIZED PERFLUOROPHENYL AZIDES - NEW REAGENTS FOR PHOTOAFFINITY-LABELING [J].

KEANA, JFW ;

CAI, SX .

JOURNAL OF FLUORINE CHEMISTRY, 1989, 43 (01) :151-154

[10] NEW REAGENTS FOR PHOTOAFFINITY-LABELING - SYNTHESIS AND PHOTOLYSIS OF FUNCTIONALIZED PERFLUOROPHENYL AZIDES [J].

KEANA, JFW ;

CAI, SX .

JOURNAL OF ORGANIC CHEMISTRY, 1990, 55 (11) :3640-3647

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