HEXAHYDRO-1H-1-PYRINDINES FROM ACID REARRANGEMENT OF 9-ALKYLIDENE-5-(M-METHOXYPHENYL)-2-METHYLMORPHANS - A NEW STRUCTURAL TYPE OF NARCOTIC-ANTAGONISTS

被引：2

作者：

AWAYA, H

MAY, EL

ACETO, MD

HARRIS, LS

SILVERTON, JV

RICE, KC

MATTSON, MV

JACOBSON, AE

机构：

[1] VIRGINIA COMMONWEALTH UNIV,MED COLL VIRGINIA,DEPT PHARMACOL,RICHMOND,VA 23298

[2] NIDDKD,CHEM LAB,BETHESDA,MD 20892

[3] NHLBI,CHEM LAB,BETHESDA,MD 20892

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1987年 / 30卷 / 05期

关键词：

D O I：

10.1021/jm00388a037

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：947 / 950

页数：4

共 25 条

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[6] PROBES FOR NARCOTIC RECEPTOR MEDIATED PHENOMENA .9. SYNTHESIS OF (+--)-(3-ALPHA,6A-ALPHA,11A-BETA)-1,3,4,5,6,11A-HEXAHYDRO-2-METHYL-2H-3,6A-METHANOBENZOFURO[2,3-CIS]AZOCIN-10-OL, AN OXIDE-BRIDGED 5-(META-HYDROXYPHENYL)MORPHAN
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[7] PROBES FOR NARCOTIC RECEPTOR MEDIATED PHENOMENA .4. SYNTHESIS OF (+--)-2,3,4,5,6,6A-HEXAHYDRO-3-METHYL-8-HYDROXY-1H-4,11B-METHANOBENZOFURO[3,2-D]AZOCINE, AN OXIDE-BRIDGED 5-(META-HYDROXYPHENYL)MORPHAN
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[J]. JOURNAL OF ORGANIC CHEMISTRY, 1984, 49 (06) : 1051 - 1056
[8] DEWEY WL, 1970, J PHARMACOL EXP THER, V175, P435
[9] DEWEY WL, 1971, J PHARMACOL EXP THER, V179, P652
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