HIGH-AFFINITY, SATURABLE [H-3]MEPYRAMINE BINDING-SITES ON RAT-LIVER PLASMA-MEMBRANE DO NOT REPRESENT HISTAMINE-H1-RECEPTORS - A WARNING

被引:26
作者
LEURS, R
BAST, A
TIMMERMAN, H
机构
关键词
D O I
10.1016/0006-2952(89)90073-7
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:2175 / 2180
页数:6
相关论文
共 17 条
[1]  
BRADFORD MM, 1976, ANAL BIOCHEM, V72, P248, DOI 10.1016/0003-2697(76)90527-3
[2]   HETEROGENEITY OF HISTAMINE H1-RECEPTORS - SPECIES VARIATIONS IN [MEPYRAMINE-H-3 BINDING OF BRAIN MEMBRANES [J].
CHANG, RSL ;
TRAN, VT ;
SNYDER, SH .
JOURNAL OF NEUROCHEMISTRY, 1979, 32 (06) :1653-1663
[3]   CORRELATION OF HISTAMINE-H1 RECEPTOR FUNCTION AND [H-3] MEPYRAMINE BINDING IN PORCINE TRACHEAL TISSUE [J].
DRIVER, AG ;
MUSTAFA, SJ .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1987, 139 (03) :287-295
[4]   SOLUBILIZATION, CHARACTERIZATION AND PARTIAL-PURIFICATION OF [H-3] MEPYRAMINE-BINDING PROTEIN, A POSSIBLE HISTAMINE H-1 RECEPTOR, FROM RAT-LIVER MEMBRANE [J].
FUKUI, H ;
WANG, NP ;
WATANABE, T ;
WADA, H .
JAPANESE JOURNAL OF PHARMACOLOGY, 1988, 46 (02) :127-139
[5]  
GARCIASAINZ JA, 1986, MOL PHARMACOL, V31, P253
[6]   SPECIFIC BINDING OF MEPYRAMINE-H-3 TO HISTAMINE H-1 RECEPTORS IN INTESTINAL SMOOTH-MUSCLE [J].
HILL, SJ ;
YOUNG, JM ;
MARRIAN, DH .
NATURE, 1977, 270 (5635) :361-362
[7]   HISTAMINE H1-RECEPTORS IN THE BRAIN OF THE GUINEA-PIG AND THE RAT - DIFFERENCES IN LIGAND-BINDING PROPERTIES AND REGIONAL DISTRIBUTION [J].
HILL, SJ ;
YOUNG, JM .
BRITISH JOURNAL OF PHARMACOLOGY, 1980, 68 (04) :687-696
[8]   HETEROCYCLIC AMINES WITH ANTIHISTAMINIC ACTIVITY [J].
HUTTRER, CP ;
DJERASSI, C ;
BEEARS, WL ;
MAYER, RL ;
SCHOLZ, CR .
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1946, 68 (10) :1999-2002
[9]   PREDOMINANCE OF HISTAMINE-H1 RECEPTORS ON LIVER PLASMA-MEMBRANE [J].
IMOTO, M ;
TSUCHIE, K ;
TANAKA, M ;
SUGIYAMA, S ;
OZAWA, T .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1985, 127 (03) :885-889
[10]   MOLECULAR-SIZE OF HISTAMINE H-1 RECEPTOR DETERMINED BY TARGET SIZE ANALYSIS [J].
KUNO, T ;
KUBO, N ;
TANAKA, C .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1985, 129 (03) :639-644