AGONIST AND ANTAGONIST BENZODIAZEPINE RECEPTOR INTERACTION INVITRO

被引:373
作者
MOHLER, H
RICHARDS, JG
机构
关键词
D O I
10.1038/294763a0
中图分类号
O [数理科学和化学]; P [天文学、地球科学]; Q [生物科学]; N [自然科学总论];
学科分类号
07 ; 0710 ; 09 ;
摘要
引用
收藏
页码:763 / 765
页数:3
相关论文
共 30 条
  • [1] INVITRO AND INVIVO INHIBITION BY ZOPICLONE OF BENZODIAZEPINE BINDING TO RODENT BRAIN RECEPTORS
    BLANCHARD, JC
    BOIREAU, A
    GARRET, C
    JULOU, L
    [J]. LIFE SCIENCES, 1979, 24 (26) : 2417 - 2420
  • [2] SPECIFIC BENZODIAZEPINE RECEPTORS IN RAT-BRAIN CHARACTERIZED BY HIGH-AFFINITY [DIAZEPAM-H-3] BINDING - (AFFINITY BINDING DIAZEPAM ANXIOLYTIC ACTIVITY BRAIN MEMBRANES REGIONAL DISTRIBUTION)
    BRAESTRUP, C
    SQUIRES, RF
    [J]. PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1977, 74 (09) : 3805 - 3809
  • [3] INFLUENCE OF GABA RECEPTOR AGONISTS AND ANTAGONISTS ON BINDING OF DIAZEPAM-H-3 TO BENZODIAZEPINE RECEPTOR
    BRILEY, MS
    LANGER, SZ
    [J]. EUROPEAN JOURNAL OF PHARMACOLOGY, 1978, 52 (01) : 129 - 132
  • [4] IS THE BENZODIAZEPINE RECEPTOR COUPLED TO A CHLORIDE ANION CHANNEL
    COSTA, T
    RODBARD, D
    PERT, CB
    [J]. NATURE, 1979, 277 (5694) : 315 - 317
  • [5] ETHYL BETA-CARBOLINE CARBOXYLATE LOWERS SEIZURE THRESHOLD AND ANTAGONIZES FLURAZEPAM-INDUCED SEDATION IN RATS
    COWEN, PJ
    GREEN, AR
    NUTT, DJ
    MARTIN, IL
    [J]. NATURE, 1981, 290 (5801) : 54 - 55
  • [6] DARRAGH A, 1981, LANCET, V2, P8
  • [7] BENZODIAZEPINE RECOGNITION SITES ON GABA RECEPTORS
    GAVISH, M
    SNYDER, SH
    [J]. NATURE, 1980, 287 (5783) : 651 - 652
  • [8] ENDOGENOUS INHIBITOR OF GABA BINDING IN MAMMALIAN BRAIN
    GREENLEE, DV
    VANNESS, PC
    OLSEN, RW
    [J]. LIFE SCIENCES, 1978, 22 (18) : 1653 - 1662
  • [9] SELECTIVE ANTAGONISTS OF BENZODIAZEPINES
    HUNKELER, W
    MOHLER, H
    PIERI, L
    POLC, P
    BONETTI, EP
    CUMIN, R
    SCHAFFNER, R
    HAEFELY, W
    [J]. NATURE, 1981, 290 (5806) : 514 - 516
  • [10] JONES BJ, BRIT J PHARM