A NEW CONVERGENT SYNTHESIS OF ALPHA-SUBSTITUTED-BETA-CARBOLINES

被引：47

作者：

ROCCA, P ^{[1
]}

MARSAIS, F ^{[1
]}

GODARD, A ^{[1
]}

QUEGUINER, G ^{[1
]}

机构：

[1] INST NATL SCI APPL ROUEN,CHIM ORGAN FINE & HETEROCYCL LAB,CNRS,URA 1429,BP 08,F-76131 MONT ST AIGNAN,FRANCE

来源：

TETRAHEDRON | 1993年 / 49卷 / 16期

关键词：

AZACARBAZOLES; ALKALOID; BORON; CARBOLINES; CROSS-COUPLING; HALOPYRIDINES; METALATION; PALLADIUM; TIN;

D O I：

10.1016/S0040-4020(01)90161-9

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

New convergent synthesis of natural alpha-substituted-beta-carbolines through metalations, cross-couplings and intramolecular substitution via (2-aminobenzene)-boronic acid, arylstannanes and ortho-fluoroiodopyridines.

引用

页码：3325 / 3342

页数：18

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