PROLONGED BLOCKADE OF OPIOID EFFECT WITH ORAL NALMEFENE

被引:58
作者
GAL, TJ [1 ]
DIFAZIO, CA [1 ]
DIXON, R [1 ]
机构
[1] KEY PHARMACEUT INC,MIAMI,FL
关键词
D O I
10.1038/clpt.1986.220
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:537 / 542
页数:6
相关论文
共 19 条
[1]  
BUSCHBAUM MS, 1977, NATURE, V270, P620
[2]   NALMEFENE - RADIOIMMUNOASSAY FOR A NEW OPIOID ANTAGONIST [J].
DIXON, R ;
HSIAO, J ;
TAAFFE, W ;
HAHN, E ;
TUTTLE, R .
JOURNAL OF PHARMACEUTICAL SCIENCES, 1984, 73 (11) :1645-1646
[3]   NALMEFENE - INTRAVENOUS SAFETY AND KINETICS OF A NEW OPIOID ANTAGONIST [J].
DIXON, R ;
HOWES, J ;
GENTILE, J ;
HSU, HB ;
HSIAO, J ;
GARG, D ;
WEIDLER, D ;
MEYER, M ;
TUTTLE, R .
CLINICAL PHARMACOLOGY & THERAPEUTICS, 1986, 39 (01) :49-53
[4]  
FISHMAN J, 1973, J PHARMACOL EXP THER, V187, P575
[5]   ANALGESIC AND RESPIRATORY DEPRESSANT ACTIVITY OF NALBUPHINE - A COMPARISON WITH MORPHINE [J].
GAL, TJ ;
DIFAZIO, CA ;
MOSCICKI, J .
ANESTHESIOLOGY, 1982, 57 (05) :367-374
[6]   PROLONGED ANTAGONISM OF OPIOID ACTION WITH INTRAVENOUS NALMEFENE IN MAN [J].
GAL, TJ ;
DIFAZIO, CA .
ANESTHESIOLOGY, 1986, 64 (02) :175-180
[7]  
GINZBURG HM, 1984, J CLIN PSYCHIAT, V45, P39
[8]   AVERSIVE EFFECTS OF NALTREXONE IN SUBJECTS NOT DEPENDENT ON OPIATES [J].
HOLLISTER, LE ;
JOHNSON, K ;
BOUKHABZA, D ;
GILLESPIE, HK .
DRUG AND ALCOHOL DEPENDENCE, 1981, 8 (01) :37-41
[9]  
JUDD LL, 1980, ARCH GEN PSYCHIAT, V37, P583
[10]  
MARTIN WR, 1973, ARCH GEN PSYCHIAT, V28, P784