TRANSFER OF ACTIVATION FROM INDOLES TO ALCOHOLS - A NEW METHOD FOR THE SYNTHESIS OF AMINOETHYLINDOLES

被引：13

作者：

EISSENSTAT, MA ^{[1
]}

WEAVER, JD ^{[1
]}

机构：

[1] STERLING WINTHROP PHARMACEUT,DIV RES,DEPT MED CHEM,COLLEGEVILLE,PA 19426

来源：

TETRAHEDRON LETTERS | 1995年 / 36卷 / 12期

关键词：

D O I：

10.1016/0040-4039(95)00229-6

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Transfer of a sulfonyl group from an indole nitrogen to a beta-amino alkoxide generates an indole anion and an aminoethylsulfonate which react to give aminoethylindoles.

引用

页码：2029 / 2032

页数：4

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