FACILE SYNTHESIS OF (+)-BREFELDIN-A

被引：42

作者：

NOKAMI, J

OHKURA, M

DANOH, Y

SAKAMOTO, Y

机构：

来源：

TETRAHEDRON LETTERS | 1991年 / 32卷 / 21期

关键词：

D O I：

10.1016/S0040-4039(00)79936-9

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

(+)-Brefeldin A (1) was synthesized by using (+)-4-cyanomethylcyclopent-2-ene-1-one (2) as a key compound. 4-Hydroxy-2-enoate functionality was built by the reaction of the aldehyde (7) with (S)-ethyl p-chlorophenylsulfinylacetate.

引用

页码：2409 / 2412

页数：4

共 22 条

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