索拉非尼的药理及临床研究

被引:15
作者
吕允凤 [1 ]
封宇飞 [2 ]
胡欣 [2 ]
毕开顺 [1 ]
机构
[1] 沈阳药科大学药物分析教研室
[2] 卫生部北京医院药学部
关键词
索拉非尼; 抗肿瘤; 多激酶抑制剂; 药理作用; 临床研究;
D O I
暂无
中图分类号
R96 [药理学];
学科分类号
100602 ; 100706 ;
摘要
索拉非尼是一种新型口服多靶点的抗肿瘤药,通过抑制Raf-1激酶从而靶向于细胞间信号传导通路直接抑制肿瘤生长,并通过抑制血管内皮生长因子受体-2(VEGF-2)和血小板衍生生长因子(PDGF)受体,阻断肿瘤血管生成途径。主要用于肾细胞癌的治疗。现综述其药理作用、药动学、临床研究、药物相互作用及不良反应的研究进展。
引用
收藏
页码:88 / 91
页数:4
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