A concise synthesis of either enantiomer of azatyrosine

被引：15

作者：

Cooper, MS ^{[1
]}

Seton, AW ^{[1
]}

Stevens, AW ^{[1
]}

Stevens, MFG ^{[1
]}

Westwell, AD ^{[1
]}

机构：

[1] UNIV NOTTINGHAM,DEPT PHARMACEUT SCI,CANC RES LABS,NOTTINGHAM NG7 2RD,ENGLAND

来源：

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS | 1996年 / 6卷 / 21期

关键词：

D O I：

10.1016/0960-894X(96)00480-5

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

A facile route to either enantiomer of azatyrosine is reported, utilising an efficient enzymic resolution of protected azatyrosine ethyl ester by alpha-chymotrypsin as a key step. Copyright (C) 1996 Elsevier Science Ltd

引用

页码：2613 / 2616

页数：4

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