The [(methyloxy)imino]methyl moiety (MOIMM) in the design of a new type of β-adrenergic blocking agent

被引：7

作者：

Balsamo, A ^{[1
]}

Macchia, M ^{[1
]}

Martinelli, A ^{[1
]}

Rossello, A ^{[1
]}

机构：

[1] Univ Pisa, Dipartimento Sci Farmaceut, I-56126 Pisa, Italy

来源：

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | 1999年 / 34卷 / 04期

关键词：

beta-adrenergic antagonists; (methyloxy)imino]methyl moiety; adrenergic drugs;

D O I：

10.1016/S0223-5234(99)80079-8

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

This article summarizes the series of studies that led to the recognition of the [(methyloxy)imino]methyl moiety (MOIMM) as a bioisoster of aryl groups in the field of beta-adrenergic blocking agents. (C) Elsevier, Paris.

引用

页码：283 / 291

页数：9

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