Studies on beta-lactam antibiotics - Synthesis and antibacterial activity of novel C-3 alkyne-substituted cephalosporins

被引：9

作者：

Barrett, D

Terasawa, T

Okuda, S

Kawabata, K

Yasuda, N

Kamimura, T

Sakane, K

Takaya, T

机构：

[1] New Drug Research Laboratories, Fujisawa Pharmaceutical Co., Ltd., Yodogawa-ku, Osaka 532

[2] Department of Process Research, Merck Research Laboratories, Rahway, NJ 07065, P.O. Box 2000

来源：

JOURNAL OF ANTIBIOTICS | 1997年 / 50卷 / 01期

关键词：

D O I：

10.7164/antibiotics.50.100

中图分类号：

Q81 [生物工程学（生物技术）]; Q93 [微生物学];

学科分类号：

071005 ; 0836 ; 090102 ; 100705 ;

摘要：

[No abstract available]

引用

页码：100 / 102

页数：3

共 9 条

[1] PALLADIUM-CATALYZED CHEMISTRY OF BETA-LACTAM VINYL TRIFLATES - COUPLING WITH ORGANOSTANNANES AND ALKOXYCARBONYLATION [J].

COOK, GK ;

HORNBACK, WJ ;

JORDAN, CL ;

MCDONALD, JH ;

MUNROE, JE .

JOURNAL OF ORGANIC CHEMISTRY, 1989, 54 (24) :5828-5830

[2]

DUERCKHEIMER W, 1985, ANGEW CHEM INT EDIT, V24, P190

[3] PALLADIUM CATALYSIS IN CEPHALOSPORIN CHEMISTRY - GENERAL METHODOLOGY FOR THE SYNTHESIS OF CEPHEM SIDE-CHAINS [J].

FARINA, V ;

BAKER, SR ;

BENIGNI, DA ;

HAUCK, SI ;

SAPINO, C .

JOURNAL OF ORGANIC CHEMISTRY, 1990, 55 (23) :5833-5847

[4] FK-482, A NEW ORALLY ACTIVE CEPHALOSPORIN SYNTHESIS AND BIOLOGICAL PROPERTIES [J].

INAMOTO, Y ;

CHIBA, T ;

KAMIMURA, T ;

TAKAYA, T .

JOURNAL OF ANTIBIOTICS, 1988, 41 (06) :828-830

[5] STUDIES ON FK482 (CEFDINIR) .4. SYNTHESIS AND STRUCTURE-ACTIVITY-RELATIONSHIPS OF 7-BETA-[(Z)-2-(2-AMINOTHIAZOL-4-YL)-2-HYDROXYIMINOACETAMIDO]-3-SUBSTITUTED CEPHALOSPORIN DERIVATIVES [J].

INAMOTO, Y ;

SAKANE, K ;

KAMIMURA, T ;

TAKAYA, T .

YAKUGAKU ZASSHI-JOURNAL OF THE PHARMACEUTICAL SOCIETY OF JAPAN, 1990, 110 (12) :908-915

[6]

KAWABATA K, 1986, J ANTIBIOT, V39, P394, DOI 10.7164/antibiotics.39.394

[7] Synthesis and biological activity of C-3 direct heterocyclylcarbon-substituted novel cephalosporins [J].

Lee, YS ;

Park, H .

JOURNAL OF ANTIBIOTICS, 1996, 49 (04) :405-407

[8]

Sakane Kazuo, 1992, Japanese Journal of Antibiotics, V45, P909

[9] STUDIES ON BETA-LACTAM ANTIBIOTICS .9. SYNTHESIS AND BIOLOGICAL-ACTIVITY OF A NEW ORALLY ACTIVE CEPHALOSPORIN, CEFIXIME (FK027) [J].

YAMANAKA, H ;

CHIBA, T ;

KAWABATA, K ;

TAKASUGI, H ;

MASUGI, T ;

TAKAYA, T .

JOURNAL OF ANTIBIOTICS, 1985, 38 (12) :1738-1751

← 1 →